SCHEMBL28795341

SCHEMBL28795341

COc1cc(N2CC(N3CCN(C(=O)OC(C)(C)C)CC3)C2)ccc1N

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.45
LMNA P02545 1/20 0.45
MAPT P10636 1/20 0.45
ALK Q9UM73 5/20 0.45
EGFR P00533 2/20 0.43
GPR119 Q8TDV5 5/20 0.43
STS P08842 1/20 0.42
PDE4B Q07343 1/20 0.42
ABCB1 P08183 2/20 0.42
SMARCA2 P51531 1/20 0.41
SMARCA4 P51532 1/20 0.41
PBRM1 Q86U86 1/20 0.41
SUV39H2 Q9H5I1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24206633 0.92 ALDH1A1 (0.45) ALDH1A1LMNAMAPTALKEGFR
SCHEMBL29803097 0.92 ALDH1A1 (0.45) ALDH1A1LMNAMAPTALKEGFR
SCHEMBL29788218 0.91 EGFR (0.52) ALDH1A1LMNAMAPTALKEGFR
SCHEMBL21133577 0.91 EGFR (0.52) ALDH1A1LMNAMAPTALKEGFR
SCHEMBL29060016 0.90 EGFR (0.51) ALDH1A1LMNAMAPTALKEGFR
SCHEMBL14406656 0.88 EGFR (0.52) ALDH1A1LMNAMAPTALKEGFR
SCHEMBL29803089 0.88 EGFR (0.52) ALDH1A1LMNAMAPTALKEGFR
SCHEMBL1707770 0.88 MAPT (0.57) ALDH1A1LMNAMAPTALKGPR119
SCHEMBL28795317 0.84 HDAC1 (0.48) ALKGPR119PDE4B
SCHEMBL28795348 0.84 ALDH1A1 (0.53) ALDH1A1LMNAMAPTALKEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114805303-A Molecule with double functions of degrading EGFR (epidermal growth factor receptor), composition and pharmaceutical application thereof 海思科医药集团股份有限公司 2022-07-29 CN disclosed