SCHEMBL28795348

SCHEMBL28795348

COc1cc(N2CC(N3CCN(C(=O)OC(C)(C)C)CC3)C2)ccc1[N+](=O)[O-]

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.53
LMNA P02545 2/20 0.53
MAPT P10636 3/20 0.52
SIRT6 Q8N6T7 1/20 0.51
ALK Q9UM73 5/20 0.42
EGFR P00533 2/20 0.42
MET P08581 1/20 0.41
KDM4E B2RXH2 1/20 0.40
CCNT1 O60563 1/20 0.40
CDK9 P50750 1/20 0.40
STS P08842 1/20 0.40
PDE4B Q07343 1/20 0.40
ABCB1 P08183 1/20 0.40
GPR119 Q8TDV5 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25370804 0.92 SIRT6 (0.56) ALDH1A1LMNAMAPTSIRT6ALK
SCHEMBL517794 0.91 ALDH1A1 (0.55) ALDH1A1LMNAMAPTSIRT6ALK
SCHEMBL310364 0.89 SIRT6 (0.55) ALDH1A1LMNAMAPTSIRT6ALK
SCHEMBL29802982 0.89 MAPT (0.65) ALDH1A1LMNAMAPTSIRT6ALK
SCHEMBL310369 0.89 MAPT (0.65) ALDH1A1LMNAMAPTSIRT6ALK
SCHEMBL310101 0.84 GPR119 (0.59) ALDH1A1LMNAMAPTSIRT6GPR119
SCHEMBL28795341 0.84 ALDH1A1 (0.45) ALDH1A1LMNAMAPTALKEGFR
SCHEMBL17411227 0.83 ALDH1A1 (0.59) ALDH1A1LMNAMAPTSIRT6ALK
SCHEMBL29986023 0.82 MAPT (0.76) ALDH1A1LMNAMAPTGPR119
SCHEMBL28945679 0.81 ALDH1A1 (0.54) ALDH1A1LMNAMAPTSIRT6ALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114805303-A Molecule with double functions of degrading EGFR (epidermal growth factor receptor), composition and pharmaceutical application thereof 海思科医药集团股份有限公司 2022-07-29 CN disclosed