SCHEMBL28795494

SCHEMBL28795494

S=C(c1cccc2nc3ccccc3cc12)c1cccc2nc3ccccc3cc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.55
KMT2A Q03164 5/20 0.55
GAA P10253 4/20 0.55
KDM4E B2RXH2 4/20 0.55
HPGD P15428 3/20 0.55
RAB9A P51151 3/20 0.55
GLA P06280 2/20 0.55
NPC1 O15118 2/20 0.55
LMNA P02545 1/20 0.55
POLB P06746 1/20 0.55
PTBP1 P26599 1/20 0.55
RCE1 Q9Y256 1/20 0.55
MAPT P10636 3/20 0.50
ACHE P22303 1/20 0.50
ESR1 P03372 2/20 0.40
ESR2 Q92731 2/20 0.40
HTR3A P46098 1/20 0.39
STAT3 P40763 1/20 0.39
NQO2 P16083 1/20 0.39
IKBKB O14920 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30075088 0.89 ALDH1A1 (0.55) ALDH1A1KMT2AGAAKDM4EHPGD
SCHEMBL28228752 0.86 ALDH1A1 (0.56) ALDH1A1KMT2AGAAKDM4EHPGD
Thiourea SCHEMBL27997998 0.82 ALDH1A1 (0.58) ALDH1A1KMT2AGAAKDM4EHPGD
SCHEMBL222908 0.81 NR4A1 (0.60) ALDH1A1KMT2AGAAKDM4EHPGD
SCHEMBL27356901 0.81 ALDH1A1 (0.55) ALDH1A1KMT2AGAAKDM4EHPGD
Water SCHEMBL7769203 0.80 NR4A1 (0.58) ALDH1A1KMT2AGAAKDM4EHPGD
SCHEMBL8850857 0.80 NR4A1 (0.58) ALDH1A1KMT2AGAAKDM4EHPGD
SCHEMBL5352931 0.80 ALDH1A1 (0.53) ALDH1A1KMT2AGAAKDM4EHPGD
Acridine SCHEMBL29774329 0.80 NR4A1 (0.58) ALDH1A1KMT2AGAAKDM4EHPGD
Acridine SCHEMBL31147690 0.80 NR4A1 (0.58) ALDH1A1KMT2AGAAKDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102231983-A Hematopoietic protection against ionizing radiation using selective cyclin-dependent kinase 4/6 inhibitors UNIV NORTH CAROLINA 2011-11-02 CN claimed
CN-102231984-A Hematopoietic protection against chemotherapeutic compounds using selective cyclin dependent kinase 4/6 inhibitors UNIV NORTH CAROLINA 2011-11-02 CN claimed
CN-103501789-A Protection of renal tissue from ischemia by inhibition of the proliferative kinases CDK4 and CDK6 UNIV NORTH CAROLINA 2014-01-08 CN disclosed
CN-102458443-A Cyclin-dependent kinase inhibitors and methods of use UNIV NORTH CAROLINA 2012-05-16 CN disclosed
CN-102231983-A Hematopoietic protection against ionizing radiation using selective cyclin-dependent kinase 4/6 inhibitors UNIV NORTH CAROLINA 2011-11-02 CN disclosed
CN-102231984-A Hematopoietic protection against chemotherapeutic compounds using selective cyclin dependent kinase 4/6 inhibitors UNIV NORTH CAROLINA 2011-11-02 CN disclosed