SCHEMBL28796567

SCHEMBL28796567

CC(=O)Oc1nc(N2CCOCC2)cc(=O)n1C.[NaH]

nearest known ligand 0.55

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 18/20 0.55
PIK3CB P42338 7/20 0.48
PIK3CD O00329 6/20 0.48
PIK3CA P42336 2/20 0.45
CYP3A4 P08684 2/20 0.45
PIK3CG P48736 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acetic Acid SCHEMBL28796568 0.76 AKT1 (0.54) AKT1PIK3CBPIK3CDPIK3CACYP3A4
SCHEMBL28796489 0.74 MEN1 (0.56) AKT1PIK3CBPIK3CDPIK3CACYP3A4
SCHEMBL1031205 0.73 AKT1 (0.72) AKT1PIK3CBPIK3CDPIK3CACYP3A4
SCHEMBL27863831 0.72 MEN1 (0.56) AKT1PIK3CBPIK3CDPIK3CACYP3A4
SCHEMBL27508637 0.71 MAPT (0.44) AKT1PIK3CB
SCHEMBL12476025 0.71 AKT1 (1.00) AKT1PIK3CBPIK3CDPIK3CACYP3A4
SCHEMBL27700148 0.69 L3MBTL1 (0.46) AKT1PIK3CB
SCHEMBL28514506 0.68 AKT1 (0.60) AKT1PIK3CBPIK3CDPIK3CACYP3A4
SCHEMBL28517851 0.67 RAF1 (0.51) AKT1PIK3CBPIK3CDPIK3CACYP3A4
SCHEMBL16742890 0.66 MAPT (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102548970-A Novel (6-oxo-1, 6-dihydropyrimidin-2-yl) amide derivatives, process for their preparation and their medical use as akt (pkb) phosphorylation inhibitors SANOFI AVENTIS 2012-07-04 CN disclosed