SCHEMBL28798652

SCHEMBL28798652

CCC(=O)c1cc(C#N)cc(C(F)(F)F)c1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.47
RXRG P48443 1/20 0.47
CES2 O00748 1/20 0.46
MRGPRX4 Q96LA9 4/20 0.43
GPBAR1 Q8TDU6 1/20 0.42
TAS2R14 Q9NYV8 1/20 0.41
RAB9A P51151 1/20 0.40
DDR1 Q08345 2/20 0.40
NOTUM Q6P988 1/20 0.39
USP2 O75604 2/20 0.38
CYP2D6 P10635 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
CTSK P43235 1/20 0.38
VNN1 O95497 1/20 0.38
PPARG P37231 1/20 0.38
PPARA Q07869 1/20 0.38
CYP2C19 P33261 1/20 0.37
TMPRSS4 Q9NRS4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29656570 1.00 RXRA (0.47) RXRARXRGCES2MRGPRX4GPBAR1
SCHEMBL5898589 0.83 CES2 (0.59) RXRARXRGCES2NOTUMPPARG
SCHEMBL2393798 0.82 CES2 (0.50) RXRARXRGCES2MRGPRX4GPBAR1
SCHEMBL29488327 0.80 MRGPRX4 (0.57) RXRARXRGCES2MRGPRX4GPBAR1
SCHEMBL545065 0.80 MRGPRX4 (0.57) RXRARXRGCES2MRGPRX4GPBAR1
SCHEMBL2789789 0.79 CES2 (0.50) RXRARXRGCES2MRGPRX4GPBAR1
SCHEMBL20646737 0.79
SCHEMBL4283632 0.79 CES2 (0.50) RXRARXRGCES2MRGPRX4GPBAR1
SCHEMBL16961681 0.78 CES2 (0.44) RXRARXRGCES2MRGPRX4GPBAR1
SCHEMBL545041 0.78 NOTUM (0.60) RXRARXRGCES2MRGPRX4GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114539245-A Pyrimidine-fused ring derivative-containing regulator, and preparation method and application thereof 上海翰森生物医药科技有限公司 2022-05-27 CN disclosed