SCHEMBL28801038

SCHEMBL28801038

O=C(NCC1CCNC1)c1ccncc1

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 5/20 0.60
SMYD3 Q9H7B4 3/20 0.55
PBK Q96KB5 5/20 0.47
USP30 Q70CQ3 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.44
KDM4E B2RXH2 1/20 0.44
MPO P05164 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
ADORA3 P0DMS8 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2A6 P11509 1/20 0.44
CYP2C19 P33261 1/20 0.44
DPP4 P27487 1/20 0.43
PREP P48147 1/20 0.43
FAP Q12884 1/20 0.43
DPP8 Q6V1X1 1/20 0.43
DPP9 Q86TI2 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13325381 0.85 NAMPT (0.63) NAMPTSMYD3SMN1; SMN2KDM4E
SCHEMBL5094284 0.85 NAMPT (0.63) NAMPTSMYD3SMN1; SMN2KDM4E
SCHEMBL13325386 0.85 NAMPT (0.63) NAMPTSMYD3SMN1; SMN2KDM4E
SCHEMBL14720114 0.83 SMYD3 (0.58) NAMPTSMYD3KDM4E
SCHEMBL17888454 0.83 SMYD3 (0.58) NAMPTSMYD3CYP2D6
SCHEMBL8255991 0.83 SMYD3 (0.58) NAMPTSMYD3
SCHEMBL21900928 0.81 NAMPT (0.59) NAMPTSMYD3
SCHEMBL17886756 0.81 SMYD3 (0.56) NAMPTSMYD3SMN1; SMN2
SCHEMBL8257484 0.80 SMN1; SMN2 (0.55) NAMPTSMYD3SMN1; SMN2
SCHEMBL8257974 0.78 SMYD3 (0.53) NAMPTSMYD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102924445-A PIM kinase inhibitor, preparation method thereof, and application thereof in pharmacy SHANGHAI JIKAI MEDICAL TECHNOLOGY CO LTD 2013-02-13 CN disclosed