SCHEMBL28801518

SCHEMBL28801518

CN(C)c1cc(C=O)cc(CCBr)c1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.41
CYP2A13 Q16696 1/20 0.41
ALDH1A1 P00352 2/20 0.32
ALDH3A1 P30838 1/20 0.32
ALDH1A3 P47895 1/20 0.32
CYP3A4 P08684 1/20 0.31
TSHR P16473 1/20 0.31
MAPK1 P28482 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
CALM1 P0DP23 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1764812 0.86 CYP2A6 (0.44) CYP2A6CYP2A13ALDH1A1ALDH3A1ALDH1A3
SCHEMBL27895303 0.84 CALM1 (0.31) CALM1
SCHEMBL12555616 0.79 CYP2A6 (0.44) CYP2A6CYP2A13ALDH1A1ALDH3A1ALDH1A3
SCHEMBL7284916 0.77 CYP2A6 (0.58) CYP2A6CYP2A13ALDH1A1ALDH3A1ALDH1A3
SCHEMBL1662928 0.77 CYP2A6 (0.58) CYP2A6CYP2A13ALDH1A1ALDH3A1ALDH1A3
SCHEMBL28781437 0.77 CYP2A6 (0.35) CYP2A6TDP1
SCHEMBL1764803 0.69 ALDH1A1 (0.30) ALDH1A1CYP3A4TSHRMAPK1TDP1
SCHEMBL5202353 0.68 CYP2A6 (0.48) CYP2A6CYP2A13ALDH1A1ALDH3A1ALDH1A3
SCHEMBL29954356 0.68 PTGS1 (0.48) CYP2A6CYP2A13ALDH1A1TSHRTDP1
SCHEMBL1764768 0.68 CYP2A6 (0.34) CYP2A6CYP2A13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102753538-B Sultam derivatives HOFFMANN LA ROCHE 2015-04-08 CN disclosed
CN-102753538-A Sultam derivatives HOFFMANN LA ROCHE 2012-10-24 CN disclosed