SCHEMBL28806387

SCHEMBL28806387

Nc1ccc(N2CCN(C=O)CC2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.57
MAPT P10636 9/20 0.57
GFER P55789 6/20 0.57
LMNA P02545 6/20 0.57
GAA P10253 5/20 0.57
KDM4E B2RXH2 4/20 0.57
HTT P42858 2/20 0.57
KMT2A Q03164 2/20 0.57
MAPK1 P28482 2/20 0.57
TDP1 Q9NUW8 2/20 0.57
ADRA2C P18825 1/20 0.57
PTK2B Q14289 1/20 0.57
ESR2 Q92731 1/20 0.57
L3MBTL1 Q9Y468 2/20 0.53
MEN1 O00255 1/20 0.53
NPC1 O15118 1/20 0.53
USP2 O75604 1/20 0.53
TP53 P04637 1/20 0.53
POLB P06746 1/20 0.53
THRB P10828 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23967058 0.84 ALDH1A1 (0.46) ALDH1A1MAPTGFERLMNAGAA
SCHEMBL6151120 0.82 MAPT (0.77) ALDH1A1MAPTGFERLMNAGAA
SCHEMBL7043679 0.82 MAPT (0.77) ALDH1A1MAPTGFERLMNAGAA
SCHEMBL23347931 0.82 MAPT (0.77) ALDH1A1MAPTGFERLMNAGAA
SCHEMBL4052281 0.81 AKR1C3 (0.52) ALDH1A1MAPTLMNAGAAKMT2A
SCHEMBL13632365 0.80 AKR1C3 (0.53) ALDH1A1MAPTGAAKDM4EKMT2A
SCHEMBL10566136 0.80 MAPT (0.52) ALDH1A1MAPTLMNAGAAKDM4E
SCHEMBL13632364 0.80 AKR1C3 (0.53) ALDH1A1MAPTLMNAKDM4EHTT
SCHEMBL5692418 0.80 TRIM24 (0.68) ALDH1A1GAAKDM4ESMN1; SMN2PDGFRB
SCHEMBL8717879 0.80 AKR1C3 (0.54) ALDH1A1MAPTLMNAGAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103435553-A Piperazine structure-based aryl formamide Raf kinase inhibitor and preparation method as well as application thereof UNIV CHINA PHARMA 2013-12-11 CN disclosed