SCHEMBL28809188

SCHEMBL28809188

Cn1cc(-c2ccc3[nH]cc(C(=O)Nc4ccncc4)c3c2)cn1

nearest known ligand 0.59

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
IKBKE Q14164 2/20 0.59
TBK1 Q9UHD2 2/20 0.59
CREBBP Q92793 2/20 0.53
GSK3B P49841 9/20 0.49
DYRK1A Q13627 9/20 0.49
CLK2 P49760 1/20 0.48
CLK3 P49761 1/20 0.48
MCL1 Q07820 1/20 0.48
WNT1 P04628 1/20 0.47
NR4A2 P43354 1/20 0.46
LRRK2 Q5S007 2/20 0.46
MET P08581 1/20 0.45
BRD4 O60885 1/20 0.45
ROCK1 Q13464 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29754046 1.00 IKBKE (0.59) IKBKETBK1CREBBPGSK3BDYRK1A
SCHEMBL28809765 0.87 IKBKE (0.51) IKBKETBK1CREBBPGSK3BDYRK1A
SCHEMBL29754042 0.87 IKBKE (0.51) IKBKETBK1CREBBPGSK3BDYRK1A
SCHEMBL29754174 0.87 GSK3B (0.50) IKBKETBK1CREBBPGSK3BDYRK1A
SCHEMBL28810262 0.87 GSK3B (0.50) IKBKETBK1CREBBPGSK3BDYRK1A
Hydrochloric Acid SCHEMBL29754051 0.82 GSK3B (0.58) GSK3BDYRK1A
Hydrochloric Acid SCHEMBL28809194 0.82 GSK3B (0.58) GSK3BDYRK1A
SCHEMBL29753969 0.82 IKBKE (0.63) IKBKETBK1GSK3BDYRK1ACLK2
SCHEMBL29754041 0.81 IKBKE (0.60) IKBKETBK1MCL1NR4A2ROCK1
SCHEMBL28809170 0.81 IKBKE (0.60) IKBKETBK1MCL1NR4A2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114867718-A Novel indazole derivative and use thereof 韩国化学研究院 2022-08-05 CN disclosed