SCHEMBL28810262

SCHEMBL28810262

CC(C)n1cc(-c2ccc3[nH]cc(C(=O)Nc4ccncc4)c3c2)cn1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.50
DYRK1A Q13627 1/20 0.50
NTRK1 P04629 1/20 0.44
IKBKE Q14164 6/20 0.44
TBK1 Q9UHD2 6/20 0.44
NR4A2 P43354 1/20 0.44
ROCK1 Q13464 2/20 0.43
MKNK1 Q9BUB5 1/20 0.43
MKNK2 Q9HBH9 1/20 0.43
PIK3CG P48736 1/20 0.41
CREBBP Q92793 1/20 0.41
NHERF1 O14745 2/20 0.41
PRMT5 O14744 1/20 0.40
WDR77 Q9BQA1 1/20 0.40
ROCK2 O75116 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29754174 1.00 GSK3B (0.50) GSK3BDYRK1ANTRK1IKBKETBK1
SCHEMBL29754046 0.87 IKBKE (0.59) GSK3BDYRK1AIKBKETBK1NR4A2
SCHEMBL28809188 0.87 IKBKE (0.59) GSK3BDYRK1AIKBKETBK1NR4A2
SCHEMBL29754042 0.83 IKBKE (0.51) GSK3BDYRK1AIKBKETBK1NR4A2
SCHEMBL28809765 0.83 IKBKE (0.51) GSK3BDYRK1AIKBKETBK1NR4A2
SCHEMBL23533876 0.82 DYRK1A (0.71) GSK3BDYRK1A
SCHEMBL28809170 0.81 IKBKE (0.60) IKBKETBK1NR4A2ROCK1NHERF1
SCHEMBL29754041 0.81 IKBKE (0.60) IKBKETBK1NR4A2ROCK1NHERF1
SCHEMBL28809217 0.79 IKBKE (0.63) GSK3BDYRK1AIKBKETBK1ROCK1
SCHEMBL29753969 0.79 IKBKE (0.63) GSK3BDYRK1AIKBKETBK1ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114867718-A Novel indazole derivative and use thereof 韩国化学研究院 2022-08-05 CN disclosed