SCHEMBL28809170

SCHEMBL28809170

O=C(Nc1ccncc1)c1c[nH]c2ccc(-c3cn[nH]c3)cc12

nearest known ligand 0.60

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
IKBKE Q14164 2/20 0.60
TBK1 Q9UHD2 2/20 0.60
ROCK2 O75116 9/20 0.53
MCL1 Q07820 2/20 0.51
NR4A2 P43354 1/20 0.50
ROCK1 Q13464 8/20 0.48
MELK Q14680 1/20 0.47
NHERF1 O14745 2/20 0.46
PRKACA P17612 1/20 0.46
PRKACG P22612 1/20 0.46
PRKACB P22694 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29754041 1.00 IKBKE (0.60) IKBKETBK1ROCK2MCL1NR4A2
SCHEMBL28810253 0.82 IKBKE (0.55) IKBKETBK1ROCK2NR4A2ROCK1
SCHEMBL29754120 0.82 IKBKE (0.55) IKBKETBK1ROCK2NR4A2ROCK1
SCHEMBL29753944 0.81 IKBKE (0.50) IKBKETBK1ROCK2NR4A2ROCK1
SCHEMBL28809197 0.81 IKBKE (0.50) IKBKETBK1ROCK2NR4A2ROCK1
SCHEMBL28809188 0.81 IKBKE (0.59) IKBKETBK1MCL1NR4A2ROCK1
SCHEMBL29754046 0.81 IKBKE (0.59) IKBKETBK1MCL1NR4A2ROCK1
SCHEMBL29754174 0.81 GSK3B (0.50) IKBKETBK1ROCK2NR4A2ROCK1
SCHEMBL28810262 0.81 GSK3B (0.50) IKBKETBK1ROCK2NR4A2ROCK1
SCHEMBL952896 0.81 DYRK1A (0.62) IKBKETBK1ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114867718-A Novel indazole derivative and use thereof 韩国化学研究院 2022-08-05 CN disclosed