SCHEMBL28809367

SCHEMBL28809367

CS(=O)(=O)c1cccc(-c2cnc(N)nc2N)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 5/20 0.58
JAK2 O60674 1/20 0.53
LOXL2 Q9Y4K0 1/20 0.50
ROCK1 Q13464 2/20 0.47
LIMK1 P53667 2/20 0.47
PTK2 Q05397 2/20 0.47
FGFR1 P11362 2/20 0.47
FLT3 P36888 2/20 0.47
AURKA O14965 1/20 0.47
DYRK3 O43781 1/20 0.47
ROCK2 O75116 1/20 0.47
PRKD3 O94806 1/20 0.47
MAP4K4 O95819 1/20 0.47
ABL1 P00519 1/20 0.47
EGFR P00533 1/20 0.47
INSR P06213 1/20 0.47
FYN P06241 1/20 0.47
CSF1R P07333 1/20 0.47
LYN P07948 1/20 0.47
KIT P10721 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL265834 0.79 CCNE2 (0.51) DHFRGSK3B
SCHEMBL264497 0.78 NPSR1 (0.51) DHFRCYP2C9
SCHEMBL4974791 0.78 DHFR (0.47) DHFR
Pyrrolidine SCHEMBL28949357 0.77 DHFR (0.52) DHFRADORA1
SCHEMBL30488016 0.77 ADORA1 (0.70) DHFRROCK1LIMK1FGFR1FLT3
SCHEMBL1388276 0.77 ADORA1 (0.70) DHFRROCK1LIMK1FGFR1FLT3
SCHEMBL6069433 0.77 RIPK2 (0.50) JAK2LOXL2ROCK1LIMK1PTK2
SCHEMBL2437223 0.77 FGFR1 (0.56) DHFRLOXL2FGFR1EGFRFYN
SCHEMBL1388358 0.77 DHFR (0.71) DHFRFGFR1MAP4K4ADORA1
SCHEMBL30401146 0.77 DHFR (0.71) DHFRFGFR1MAP4K4ADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107530430-A AGENT FOR PREVENTING AND/OR TREATING AMYOTROPHIC LATERAL SCLEROSIS 国立大学法人京都大学 2018-01-02 CN disclosed
CN-103626742-A Bi-aryl meta-pyrimidine inhibitors of kinases TARGEGEN INC 2014-03-12 CN disclosed