SCHEMBL28809441

SCHEMBL28809441

C[C@@H](c1ccccc1)n1cccc1C(N)=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
GABRA1 P14867 3/20 0.44
MAPK1 P28482 1/20 0.43
CYP1A2 P05177 3/20 0.42
CYP3A4 P08684 3/20 0.42
GABRB2 P47870 2/20 0.42
CYP11B1 P15538 2/20 0.42
CYP11B2 P19099 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
LMNA P02545 2/20 0.42
ABCB11 O95342 1/20 0.42
GABRA2 P47869 1/20 0.42
ALOX5 P09917 1/20 0.41
ADRA1D P25100 1/20 0.41
BRD4 O60885 1/20 0.40
CYP2D6 P10635 1/20 0.39
MAP3K14 Q99558 1/20 0.39
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1051047 0.86 TDP1 (0.59) ALDH1A1TDP1GABRA1MAPK1CYP1A2
SCHEMBL1051049 0.86 TDP1 (0.59) ALDH1A1TDP1GABRA1MAPK1CYP1A2
SCHEMBL24967421 0.85 ALDH1A1 (0.50) ALDH1A1TDP1GABRA1MAPK1CYP1A2
SCHEMBL19063220 0.83 ALDH1A1 (0.49) ALDH1A1TDP1GABRA1MAPK1CYP1A2
SCHEMBL24966942 0.81 MAPK1 (0.62) ALDH1A1TDP1GABRA1MAPK1CYP1A2
SCHEMBL24966945 0.81 ALDH1A1 (0.47) ALDH1A1TDP1GABRA1MAPK1CYP1A2
SCHEMBL24967609 0.81 ALDH1A1 (0.47) ALDH1A1TDP1GABRA1MAPK1CYP1A2
SCHEMBL6796081 0.80 LMNA (0.40) TDP1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL14803831 0.79 ALDH1A1 (0.44) ALDH1A1TDP1GABRA1MAPK1CYP1A2
SCHEMBL24967014 0.78 MAPK1 (0.49) ALDH1A1TDP1GABRA1MAPK1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103649089-A Pyrrolotriazinones as PI3K inhibitors ALMIRALL SA 2014-03-19 CN disclosed