SCHEMBL28810302

SCHEMBL28810302

NC(=S)CCCNC(=O)O

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PRMT1 Q99873 1/20 0.35
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
ADRA1A P35348 1/20 0.33
ATM Q13315 1/20 0.32
PLA2G4A P47712 1/20 0.32
CYP1A2 P05177 1/20 0.31
EPHX2 P34913 2/20 0.31
KDM4E B2RXH2 1/20 0.31
MAPK1 P28482 1/20 0.31
HIF1A Q16665 1/20 0.31
LMNA P02545 1/20 0.31
FABP4 P15090 1/20 0.31
PAOX Q6QHF9 2/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1493634 0.86
SCHEMBL15328337 0.79 MEN1 (0.36) PRMT1CA1CA2ADRA1AEPHX2
SCHEMBL5120839 0.79 MEN1 (0.41) PRMT1CA1CA2ADRA1AKDM4E
SCHEMBL5128168 0.77 KDM4E (0.41) PRMT1CA1CA2ADRA1AEPHX2
SCHEMBL13731191 0.76 PRMT1 (0.48) PRMT1CA1CA2ADRA1AKDM4E
SCHEMBL320940 0.75 PRMT1 (0.58) PRMT1ADRA1AATMPLA2G4AEPHX2
SCHEMBL11213979 0.75 CASP2 (0.60) MEN1KMT2A
SCHEMBL28945607 0.74 PRMT1 (0.52) PRMT1ADRA1AKDM4EMAPK1HIF1A
SCHEMBL27130042 0.74 PRMT1 (0.52) PRMT1ADRA1AKDM4EMAPK1HIF1A
SCHEMBL8958360 0.74 KDM4E (0.43) PRMT1CA1CA2ADRA1AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114746419-A N- (3- (5- (pyrimidin-4-yl) thiazol-4-yl) phenyl) sulfonamide compounds and their use as BRAF inhibitors 国家医疗保健研究所 2022-07-12 CN disclosed