SCHEMBL28810673

SCHEMBL28810673

O=C(O)n1ccc2c(F)cc(Cl)nc21

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 3/20 0.34
KEAP1 Q14145 1/20 0.33
NFE2L2 Q16236 1/20 0.33
HDAC4 P56524 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
PARP1 P09874 1/20 0.31
GRM2 Q14416 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MAOB P27338 1/20 0.30
NOTUM Q6P988 2/20 0.30
GPR35 Q9HC97 1/20 0.30
ENPP3 O14638 1/20 0.30
ENPP1 P22413 1/20 0.30
SLC22A6 Q4U2R8 1/20 0.30
ABCG2 Q9UNQ0 1/20 0.30
USP2 O75604 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23147760 0.82 KDM4E (0.36) SLC22A12HDAC4HDAC1HDAC6KDM4E
SCHEMBL29721744 0.82 KDM4E (0.36) SLC22A12HDAC4HDAC1HDAC6KDM4E
SCHEMBL28809773 0.76 SLC22A12 (0.33) SLC22A12KEAP1NFE2L2PARP1KDM4E
SCHEMBL21617815 0.72 DAO (0.39) SLC22A12KDM4ENOTUMENPP3ENPP1
SCHEMBL28881483 0.71 PARP1 (0.44) SLC22A12PARP1SLC22A6ABCG2
SCHEMBL20765651 0.70 ENPP3 (0.39) SLC22A12PARP1ENPP3ENPP1SLC22A6
SCHEMBL24843610 0.70
SCHEMBL27171964 0.68 ELANE (0.40) SLC22A12PARP1KDM4ESLC22A6ABCG2
SCHEMBL28809800 0.68
SCHEMBL23148094 0.68

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114746090-A Azaindole carboxamide compounds for the treatment of mycobacterial infections 结核病药物开发全球联盟公司 2022-07-12 CN disclosed