SCHEMBL28811925

SCHEMBL28811925

COc1ccc(C=CNC(=O)Cc2cccc3ccccc23)cc1OC

nearest known ligand 0.69

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TRPM5 Q9NZQ8 1/20 0.69
CYP3A4 P08684 1/20 0.55
CYP2D6 P10635 1/20 0.55
MAPT P10636 1/20 0.55
CYP2C9 P11712 1/20 0.55
CYP2C19 P33261 1/20 0.55
GAA P10253 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.52
ATM Q13315 2/20 0.52
KMT2A Q03164 2/20 0.52
ABCG2 Q9UNQ0 2/20 0.50
AKR1C2 P52895 1/20 0.49
BACE1 P56817 1/20 0.48
ALDH1A1 P00352 1/20 0.48
NFE2L2 Q16236 1/20 0.48
MEN1 O00255 1/20 0.47
SMPD1 P17405 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28796994 0.85 MAPT (0.58) TRPM5CYP3A4CYP2D6MAPTCYP2C9
SCHEMBL28796967 0.85 MAPT (0.58) TRPM5CYP3A4CYP2D6MAPTCYP2C9
SCHEMBL27882241 0.82 KMT2A (0.66) CYP3A4CYP2D6MAPTCYP2C9CYP2C19
SCHEMBL31612234 0.81 TRPM5 (1.00) TRPM5CYP3A4MAPTCYP2C9CYP2C19
SCHEMBL3861202 0.81 TRPM5 (1.00) TRPM5CYP3A4MAPTCYP2C9CYP2C19
SCHEMBL3861198 0.81 TRPM5 (1.00) TRPM5CYP3A4MAPTCYP2C9CYP2C19
SCHEMBL27865858 0.75 CYP3A4 (0.70) CYP3A4CYP2D6MAPTCYP2C9CYP2C19
SCHEMBL4253934 0.74 PTPN1 (0.73) TRPM5CYP3A4MAPTCYP2C19ATM
SCHEMBL9050603 0.73 L3MBTL1 (0.61) TRPM5CYP3A4CYP2D6MAPTCYP2C19
SCHEMBL3855392 0.73 BACE1 (0.74) CYP3A4CYP2D6MAPTCYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102603553-B Compound with collaborative antifungal effect and application thereof in pharmaceuticals UNIV PLA 2ND MILITARY MEDICAL 2014-07-30 CN disclosed