SCHEMBL28812840

SCHEMBL28812840

CC(=O)Oc1cccc2[nH]cc(C=O)c12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.53
SLC22A6 Q4U2R8 1/20 0.51
IMPDH2 P12268 1/20 0.42
TLR2 O60603 1/20 0.41
ERN1 O75460 1/20 0.41
TLR1 Q15399 1/20 0.41
TLR6 Q9Y2C9 1/20 0.41
MTNR1A P48039 1/20 0.40
MTNR1B P49286 1/20 0.40
MAPK1 P28482 1/20 0.39
KDM4E B2RXH2 3/20 0.38
ALDH1A1 P00352 2/20 0.38
BLM P54132 2/20 0.38
TDP1 Q9NUW8 2/20 0.38
HSD17B10 Q99714 2/20 0.38
ESR1 P03372 1/20 0.38
ITGB3 P05106 1/20 0.38
ITGA2B P08514 1/20 0.38
HMGB1 P09429 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17422040 0.87 CYP2A6 (0.54) CYP2A6SLC22A6IMPDH2TLR2ERN1
SCHEMBL8799039 0.86 CYP2A6 (0.50) CYP2A6IMPDH2TLR2ERN1TLR1
SCHEMBL1337138 0.81 CYP2A6 (0.58) CYP2A6IMPDH2TLR2ERN1TLR1
SCHEMBL29955729 0.81 CYP2A6 (0.58) CYP2A6IMPDH2TLR2ERN1TLR1
SCHEMBL15322953 0.80 BCHE (0.51) CYP2A6ACHE
SCHEMBL30297980 0.80 VCP (0.45) SLC22A6TLR2MTNR1AMTNR1BMAPK1
SCHEMBL27095369 0.79 MTNR1A (0.49) SLC22A6MTNR1AMTNR1BKDM4EALDH1A1
SCHEMBL25792506 0.79 SLC22A6 (0.58) SLC22A6MTNR1AMTNR1BMAPK1KDM4E
SCHEMBL17422135 0.78 SMN1; SMN2 (0.55) CYP2A6ALDH1A1TDP1HPGDTSHR
SCHEMBL29950589 0.78 CYP2A6 (0.54) CYP2A6IMPDH2MAPK1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103772395-A Tricyclic indole compound (I) with PARP (Poly-ADP-Ribose Polymerase) inhibiting activity, preparation method and application thereof UNIV CHINA PHARMA 2014-05-07 CN disclosed