SCHEMBL28812970

SCHEMBL28812970

O=C(c1onc(-c2ccccn2)c1C(F)(F)F)c1onc(-c2ccccn2)c1C(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 4/20 0.43
S1PR3 Q99500 3/20 0.43
HDAC4 P56524 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
GABRA5 P31644 4/20 0.39
TRPV1 Q8NER1 1/20 0.38
F2 P00734 1/20 0.38
F12 P00748 1/20 0.38
HTT P42858 1/20 0.37
HSD17B10 Q99714 1/20 0.37
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
CYP1A2 P05177 1/20 0.36
POLB P06746 1/20 0.36
CCR1 P32246 1/20 0.36
CCR5 P51681 1/20 0.36
CCR8 P51685 1/20 0.36
METAP1 P53582 1/20 0.36
BLM P54132 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL408682 0.90 S1PR1 (0.45) S1PR1S1PR3HDAC4HDAC1HDAC6
SCHEMBL405411 0.82 LMNA (0.45) S1PR1S1PR3HDAC4HDAC6GABRA5
SCHEMBL27971853 0.79 ESR1 (0.46) S1PR1S1PR3HSD17B10MEN1ALDH1A1
SCHEMBL27837002 0.76 ESR1 (0.41) S1PR1S1PR3HDAC4HDAC1HDAC6
SCHEMBL409574 0.75 PTPN1 (0.46) GABRA5HSD17B10KDM4ELMNACYP1A2
SCHEMBL27971825 0.74 GHSR (0.39) HDAC1HDAC6HSD17B10MEN1KMT2A
SCHEMBL408632 0.73 HDAC4 (0.41) S1PR1S1PR3HDAC4HDAC1HDAC6
SCHEMBL404322 0.73 PTPN1 (0.43) S1PR1S1PR3HDAC4HDAC1HDAC6
SCHEMBL27971675 0.72 PTPN5 (0.40) KDM4EALDH1A1
SCHEMBL27971673 0.72 GPBAR1 (0.45) HDAC4HDAC1HDAC6TRPV1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104030998-A 4- perfluoroalkyl-4,5-disubstituted isoxazole derivative and preparation method thereof UNIV EAST CHINA NORMAL 2014-09-10 CN claimed
CN-104030998-B 4-Polyfluoroalkyl-4,5-bis-substituted isoxazoles derivative and preparation method thereof EAST CHINA NORMAL UNIVERSITY (CN) 2015-11-18 CN disclosed
CN-104030998-A 4- perfluoroalkyl-4,5-disubstituted isoxazole derivative and preparation method thereof UNIV EAST CHINA NORMAL 2014-09-10 CN disclosed