SCHEMBL28815162

SCHEMBL28815162

CC(=O)Oc1cc(O)c2cccc(F)c2n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.42
MAPT P10636 2/20 0.42
TP53 P04637 1/20 0.42
GAA P10253 1/20 0.42
HTT P42858 1/20 0.42
HSD17B10 Q99714 1/20 0.42
GRM2 Q14416 1/20 0.39
CYP3A4 P08684 2/20 0.37
AURKA O14965 1/20 0.37
ADORA2A P29274 7/20 0.36
ADORA1 P30542 3/20 0.36
LMNA P02545 2/20 0.34
DAO P14920 1/20 0.34
DDO Q99489 1/20 0.34
TNKS O95271 1/20 0.34
PARP1 P09874 1/20 0.34
TNKS2 Q9H2K2 1/20 0.34
ALOX12 P18054 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27987879 0.79 CYP4F2 (0.38) KDM4EMAPTTP53GAAHTT
SCHEMBL2222961 0.74 ADORA2A (0.47) KDM4EMAPTTP53GAAHSD17B10
SCHEMBL22084269 0.73 KDM4E (0.42) KDM4EMAPTTP53GAAHTT
SCHEMBL1832253 0.73 CYP1A2 (0.41) KDM4EMAPTGAAHSD17B10LMNA
SCHEMBL3333164 0.73 GRM2 (0.48) KDM4EMAPTGRM2AURKAADORA2A
SCHEMBL8134178 0.71 HTT (0.39) KDM4EMAPTTP53GAAHTT
SCHEMBL27863966 0.71 ABCB11 (0.39) KDM4EMAPTTP53GAAHTT
SCHEMBL2518688 0.70 KDM4E (0.46) KDM4EMAPTGAAHSD17B10CYP3A4
SCHEMBL28815163 0.70 KDM4E (0.41) KDM4EGAAHSD17B10GRM2AURKA
SCHEMBL27988221 0.70 CYP4F2 (0.37) GAATNKSPARP1TNKS2CYP4F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102651970-B Quinoline amide m1 receptor positive allosteric modulators MERCK SHARP & DOHME 2014-11-12 CN disclosed