SCHEMBL28816299

SCHEMBL28816299

CCOC(=O)c1nc(-c2ccco2)no1

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.57
PKM P14618 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.56
HTT P42858 1/20 0.56
DAGLA Q9Y4D2 1/20 0.51
ADORA3 P0DMS8 13/20 0.50
ADORA2A P29274 12/20 0.50
ADORA1 P30542 11/20 0.50
ADORA2B P29275 5/20 0.50
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
ALOX15 P16050 1/20 0.46
HSD17B10 Q99714 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
TSHR P16473 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2163538 0.86 DAGLA (0.52) ALDH1A1PKML3MBTL1HTTDAGLA
SCHEMBL2554648 0.79 HTT (0.67) ALDH1A1HTTMEN1KMT2AHSD17B10
SCHEMBL3233714 0.76 HTT (0.71) ALDH1A1PKML3MBTL1HTTMEN1
SCHEMBL4528391 0.75 HTT (0.66) ALDH1A1HTTMEN1KMT2A
SCHEMBL1179214 0.75 ALDH1A1 (0.60) ALDH1A1PKML3MBTL1HTTMEN1
SCHEMBL28816256 0.75 MAPT (0.64) ALDH1A1PKMHTTDAGLAKMT2A
SCHEMBL8593668 0.74 HTT (0.68) ALDH1A1HTTMEN1KMT2ATSHR
SCHEMBL3335119 0.74 HTT (0.72) ALDH1A1L3MBTL1HTTHSD17B10
SCHEMBL3230760 0.74 HTT (0.68) ALDH1A1HTTMEN1KMT2ATSHR
SCHEMBL28816280 0.74 HTT (0.68) ALDH1A1PKML3MBTL1HTTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114933573-A 3-substituted-1, 2, 4-oxadiazole-5-carboxylic acid derivative, and preparation method and application thereof 贵州大学 2022-08-23 CN claimed
CN-114933573-B 3-substituted-1, 2, 4-oxadiazole-5-carboxylic acid derivative, and preparation method and application thereof 贵州大学 2023-10-20 CN disclosed
CN-114933573-A 3-substituted-1, 2, 4-oxadiazole-5-carboxylic acid derivative, and preparation method and application thereof 贵州大学 2022-08-23 CN disclosed