SCHEMBL28816669

SCHEMBL28816669

CCOC(=O)c1ocnc1CCBr

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 1/20 0.39
HSP90AA1 P07900 1/20 0.37
L3MBTL1 Q9Y468 2/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
ALDH1A1 P00352 2/20 0.35
TSHR P16473 1/20 0.35
PDE4D Q08499 1/20 0.35
KDM4E B2RXH2 2/20 0.35
AHR P35869 1/20 0.35
NPC1 O15118 1/20 0.35
MAPT P10636 1/20 0.35
RAB9A P51151 1/20 0.35
HPGD P15428 1/20 0.34
POLB P06746 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13545979 0.88 PLK1 (0.43) PLK1HSP90AA1L3MBTL1CYP1A2CYP2C9
SCHEMBL2567865 0.84 CYP1A2 (0.40) HSP90AA1L3MBTL1CYP1A2CYP2C9CYP2C19
SCHEMBL23635692 0.80 CA12 (0.38) L3MBTL1CYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL3714376 0.78 CYP1A2 (0.40) PLK1L3MBTL1CYP1A2CYP2C9CYP2C19
SCHEMBL2139059 0.77 ALDH1A1 (0.48) L3MBTL1CYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL29620241 0.76 KDM4E (0.41) CYP1A2CYP2C9CYP2C19ALDH1A1TSHR
SCHEMBL25368994 0.76 CYP1A2 (0.41) L3MBTL1CYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL22952394 0.75 ALDH1A1 (0.43) HSP90AA1L3MBTL1CYP1A2CYP2C9CYP2C19
SCHEMBL21854494 0.75 GLP1R (0.46) L3MBTL1CYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL15919895 0.74 KDM4E (0.49) HSP90AA1CYP1A2CYP2C9CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114630822-A Biaryl dihydroorotate dehydrogenase inhibitors 詹森生物科技公司 2022-06-14 CN disclosed