SCHEMBL28819563

SCHEMBL28819563

COc1ccc2nc(-c3ccc(Cl)c(Cl)c3)n(C(C(N)=O)(C3CCCC3)C3CCCC3)c2c1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 1/20 0.45
MAPK10 P53779 4/20 0.44
HCRTR1 O43613 2/20 0.41
HCRTR2 O43614 2/20 0.41
EGFR P00533 3/20 0.38
KDM4E B2RXH2 1/20 0.37
MAP3K14 Q99558 3/20 0.37
CYP11B1 P15538 1/20 0.37
CYP11B2 P19099 1/20 0.37
KMT2A Q03164 1/20 0.36
ALOX5AP P20292 1/20 0.35
CNR2 P34972 1/20 0.35
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
CCR2 P41597 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28819601 0.99 NR1H4 (0.46) NR1H4MAPK10HCRTR1HCRTR2EGFR
SCHEMBL28819648 0.86 NR1H4 (0.45) NR1H4MAPK10HCRTR1HCRTR2CYP11B1
SCHEMBL28819675 0.84 MCHR1 (0.44) NR1H4MAPK10MAP3K14
SCHEMBL28819631 0.82 CNR2 (0.45) NR1H4MAPK10KDM4EALOX5APCNR2
SCHEMBL28819698 0.82 PLA2G2A (0.42) NR1H4CYP11B1CYP11B2CNR2
SCHEMBL28948676 0.81 NR1H4 (0.40) NR1H4MAPK10CYP11B1CYP11B2ALOX5AP
SCHEMBL28819665 0.80 POLB (0.40) NR1H4MAPK10KDM4EKMT2AALOX5AP
Hydrochloric Acid SCHEMBL4213341 0.79 CNR2 (0.49) KDM4EKMT2ACNR2MAOAMAOB
Hydrochloric Acid SCHEMBL4216436 0.79 MCHR1 (0.46) ALOX5APCNR2
Hydrochloric Acid SCHEMBL4213337 0.78 CNR2 (0.48) KDM4EKMT2ACNR2MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110404073-B Methods and pharmaceutical compositions for treating hepatitis B virus infection 国家医疗保健研究所 2022-08-16 CN disclosed