SCHEMBL28820188

SCHEMBL28820188

CC(C)(C)NC(=O)O[C@@H](Cc1ccccc1)C(O)C#N

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSL P07711 5/20 0.44
CTSK P43235 5/20 0.44
CTSB P07858 4/20 0.44
SCN9A Q15858 1/20 0.44
CTSS P25774 5/20 0.44
ANPEP P15144 2/20 0.39
CTSC P53634 4/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
CTSH P09668 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27485822 0.84 SCN9A (0.47) CTSLCTSKCTSBSCN9ACTSS
SCHEMBL28020483 0.81 SCN9A (0.45) CTSLCTSKCTSBSCN9ACTSS
SCHEMBL28837742 0.81 SCN9A (0.47) CTSLCTSKCTSBSCN9ACTSS
SCHEMBL28837747 0.81 SCN9A (0.47) CTSLCTSKCTSBSCN9ACTSS
SCHEMBL28496647 0.78 CTSC (0.44) CTSLCTSKCTSBANPEPCTSC
SCHEMBL28529219 0.78 CTSC (0.44) CTSLCTSKCTSBANPEPCTSC
SCHEMBL5393871 0.77 OPRM1 (0.45) SCN9ANPC1RAB9AMAPT
SCHEMBL5393866 0.77 OPRM1 (0.45) SCN9ANPC1RAB9AMAPT
SCHEMBL28755814 0.76 CYP3A4 (0.42) SCN9A
SCHEMBL28020511 0.75 SCN9A (0.43) SCN9ARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104837858-A Ketoamide immunoproteasome inhibitors HOFFMANN LA ROCHE 2015-08-12 CN disclosed