SCHEMBL28824499

SCHEMBL28824499

COc1cccc(-c2ncccc2OC)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK4 Q9HAZ1 2/20 0.62
DYRK1A Q13627 1/20 0.62
KCNA5 P22460 1/20 0.52
AURKA O14965 1/20 0.50
PDGFRB P09619 1/20 0.49
PDGFRA P16234 1/20 0.49
TOP1 P11387 1/20 0.48
CYP19A1 P11511 1/20 0.47
PDE10A Q9Y233 2/20 0.46
PDE4B Q07343 1/20 0.46
NPY5R Q15761 1/20 0.46
CCNB2 O95067 1/20 0.46
CDK1 P06493 1/20 0.46
CCNB1 P14635 1/20 0.46
GSK3A P49840 1/20 0.46
GSK3B P49841 1/20 0.46
CDK5 Q00535 1/20 0.46
CDK5R1 Q15078 1/20 0.46
CCNB3 Q8WWL7 1/20 0.46
ABCG2 Q9UNQ0 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4049358 0.84 DYRK1A (0.51) CLK4DYRK1AKCNA5AURKAPDE4B
SCHEMBL10094648 0.83 DYRK1A (0.62) CLK4DYRK1AKCNA5AURKATOP1
SCHEMBL15674640 0.82 PDE4B (0.53) KCNA5PDE10APDE4BPDE7APDE3A
SCHEMBL7230871 0.82 MAP4K4 (0.50) CDK5CDK5R1CYP3A4ALDH1A1NPC1
SCHEMBL15674440 0.82 PDGFRB (0.51) CLK4PDGFRBPDGFRAPDE4BGSK3B
SCHEMBL27866855 0.82 DYRK1A (0.60) CLK4DYRK1AKCNA5AURKATOP1
SCHEMBL27265882 0.82 DYRK1A (0.60) CLK4DYRK1AKCNA5AURKATOP1
SCHEMBL987247 0.80 SYK (0.51) PDGFRBPDGFRAPDE3ALMNAKDM4E
SCHEMBL16047508 0.80 KCNA5 (0.62) CLK4DYRK1AKCNA5AURKATOP1
SCHEMBL10094501 0.80 DYRK1A (0.57) CLK4DYRK1AKCNA5AURKATOP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105051044-A Compounds and their use for modulating hemoglobin GLOBAL BLOOD THERAPEUTICS INC 2015-11-11 CN disclosed