SCHEMBL4049358

SCHEMBL4049358

COc1cccc(-c2ncccc2OC(C)=O)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.51
CLK4 Q9HAZ1 1/20 0.51
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
ALDH1A1 P00352 3/20 0.46
KDM4E B2RXH2 2/20 0.46
HPGD P15428 1/20 0.46
KCNA5 P22460 1/20 0.46
GAPDH P04406 1/20 0.46
PDE4A P27815 2/20 0.45
PDE4B Q07343 2/20 0.45
PDE4C Q08493 2/20 0.45
PDE4D Q08499 2/20 0.45
HTT P42858 3/20 0.45
PKM P14618 2/20 0.45
SYK P43405 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
BACE1 P56817 1/20 0.44
ADORA3 P0DMS8 2/20 0.44
ADORA2B P29275 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28824499 0.84 CLK4 (0.62) DYRK1ACLK4ALDH1A1KDM4EHPGD
SCHEMBL27504690 0.82 MAP4K4 (0.44) MEN1KMT2AALDH1A1KDM4EHPGD
SCHEMBL6717844 0.82 ALDH1A1 (0.48) ALDH1A1KDM4EHPGDHTTL3MBTL1
SCHEMBL4052629 0.79 GAPDH (0.46) MEN1KMT2AALDH1A1HPGDGAPDH
SCHEMBL27489306 0.78 PDE4D (0.55) ALDH1A1KDM4EPDE4APDE4BPDE4C
SCHEMBL22160863 0.78 DHODH (0.59) DYRK1ACLK4MEN1KMT2AALDH1A1
SCHEMBL30832877 0.78 DHODH (0.59) DYRK1ACLK4MEN1KMT2AALDH1A1
SCHEMBL24313994 0.77 HTT (0.56) ALDH1A1KDM4EGAPDHHTTPKM
SCHEMBL6174210 0.77 JAK2 (0.56) DYRK1ACLK4MEN1KMT2AKDM4E
SCHEMBL26009136 0.76 LMNA (0.59) ALDH1A1GAPDHHTTBACE1ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2024371-A1 PHENANTHRENE DERIVATIVES AS MPGES-1 INHIBITORS Merck Frosst Canada Ltd. (CA) 2009-02-18 EP disclosed
WO-2007134434-A1 PHENANTHRENE DERIVATIVES AS MPGES-1 INHIBITORS MERCK FROSST CANADA LTD. (CA) 2007-11-29 WO disclosed