SCHEMBL28825474

SCHEMBL28825474

COc1ncccc1Cn1ccc(-c2ccc(OC(F)F)c(F)c2)n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 4/20 0.51
GRIN1 Q05586 3/20 0.51
SMN1; SMN2 Q16637 3/20 0.40
NPC1 O15118 2/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
GLA P06280 1/20 0.40
GAA P10253 1/20 0.40
HPGD P15428 1/20 0.40
RAB9A P51151 1/20 0.40
P2RX3 P56373 1/20 0.39
PDE1A P54750 1/20 0.39
PDE1B Q01064 1/20 0.39
PDE1C Q14123 1/20 0.39
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
RXRA P19793 1/20 0.37
ALOX5AP P20292 1/20 0.37
FEN1 P39748 1/20 0.37
MET P08581 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28825641 0.86 GRIN1 (0.50) GRIN2BGRIN1SMN1; SMN2NPC1KDM4E
SCHEMBL28825521 0.78 GRIN2B (0.51) GRIN2BGRIN1SMN1; SMN2NPC1KDM4E
SCHEMBL28825542 0.77 GRIN2B (0.51) GRIN2BGRIN1P2RX3
SCHEMBL28825452 0.77 GRIN2B (0.50) GRIN2BGRIN1SMN1; SMN2NPC1KDM4E
SCHEMBL28964555 0.77 GRIN2B (0.49) GRIN2BGRIN1SMN1; SMN2NPC1KDM4E
SCHEMBL28825469 0.76 GRIN2B (0.49) GRIN2BGRIN1SMN1; SMN2NPC1KDM4E
SCHEMBL28949594 0.76 MAPT (0.44) GRIN2BGRIN1SMN1; SMN2NPC1KDM4E
SCHEMBL28825488 0.75 GRIN2B (0.50) GRIN2BGRIN1
SCHEMBL28825586 0.75 GRIN2B (0.48) GRIN2BGRIN1PDE4D
SCHEMBL28825649 0.73 GRIN2B (0.47) GRIN2BGRIN1SMN1; SMN2NPC1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN claimed
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN disclosed