SCHEMBL28825632

SCHEMBL28825632

Cc1cncc(Cn2ccc(-c3ccc(C(C)(F)F)cc3)n2)c1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
HTT P42858 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
GRIN1 Q05586 9/20 0.44
GRIN2B Q13224 9/20 0.44
KDM1A O60341 2/20 0.40
HDAC1 Q13547 2/20 0.40
CYP11B1 P15538 4/20 0.39
CYP11B2 P19099 4/20 0.39
TDP1 Q9NUW8 2/20 0.38
MAPT P10636 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
KDM4E B2RXH2 1/20 0.38
NPC1 O15118 1/20 0.38
LMNA P02545 1/20 0.38
HPGD P15428 1/20 0.38
RAB9A P51151 1/20 0.38
CYP3A4 P08684 1/20 0.36
NR3C1 P04150 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28949591 0.88 ALDH1A1 (0.44) ALDH1A1HTTNPSR1GRIN1GRIN2B
SCHEMBL28825495 0.84 GRIN1 (0.47) ALDH1A1HTTNPSR1GRIN1GRIN2B
SCHEMBL28825651 0.81 GRIN1 (0.52) ALDH1A1HTTNPSR1GRIN1GRIN2B
SCHEMBL28825484 0.80 GRIN1 (0.43) ALDH1A1HTTNPSR1GRIN1GRIN2B
SCHEMBL28949596 0.79 GRIN1 (0.42) ALDH1A1GRIN1GRIN2BKDM1AHDAC1
SCHEMBL26192810 0.78 CYP11B1 (0.48) ALDH1A1NPSR1GRIN1GRIN2BCYP11B1
SCHEMBL28825551 0.76 GRIN2B (0.47) ALDH1A1GRIN1GRIN2BKDM1AHDAC1
SCHEMBL28825494 0.74 GRIN2B (0.46) ALDH1A1HTTNPSR1GRIN1GRIN2B
SCHEMBL28825489 0.73 GRIN2B (0.48) GRIN1GRIN2B
SCHEMBL28825543 0.73 GRIN2B (0.48) ALDH1A1HTTNPSR1GRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN claimed
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN disclosed