SCHEMBL28825484

SCHEMBL28825484

Cc1cncc(Cn2ccc(-c3ccc(C)c(F)c3)n2)c1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 13/20 0.43
GRIN2B Q13224 13/20 0.43
KCNH2 Q12809 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
MAPT P10636 1/20 0.40
KDM1A O60341 2/20 0.40
HDAC1 Q13547 2/20 0.40
MEN1 O00255 1/20 0.39
NPC1 O15118 1/20 0.39
KMT2A Q03164 1/20 0.39
ALDH1A1 P00352 1/20 0.38
HTT P42858 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28825651 0.91 GRIN1 (0.52) GRIN1GRIN2BSMN1; SMN2MAPTKDM1A
SCHEMBL28825507 0.90 SMN1; SMN2 (0.45) GRIN1GRIN2BKCNH2SMN1; SMN2MAPT
SCHEMBL28949596 0.88 GRIN1 (0.42) GRIN1GRIN2BSMN1; SMN2MAPTKDM1A
SCHEMBL28825551 0.86 GRIN2B (0.47) GRIN1GRIN2BKCNH2SMN1; SMN2MAPT
SCHEMBL28825495 0.85 GRIN1 (0.47) GRIN1GRIN2BKCNH2SMN1; SMN2MAPT
SCHEMBL28825489 0.83 GRIN2B (0.48) GRIN1GRIN2BKCNH2
SCHEMBL28825580 0.81 GRIN1 (0.43) GRIN1GRIN2BKCNH2SMN1; SMN2MAPT
SCHEMBL28825632 0.80 ALDH1A1 (0.44) GRIN1GRIN2BSMN1; SMN2MAPTKDM1A
SCHEMBL26192810 0.79 CYP11B1 (0.48) GRIN1GRIN2BSMN1; SMN2MAPTMEN1
SCHEMBL28825447 0.79 GRIN2B (0.50) GRIN1GRIN2BSMN1; SMN2MAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN claimed
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN disclosed