SCHEMBL28825820

SCHEMBL28825820

COc1ccc(CN2CC(C)(C)c3ccc(C(C)=O)cc32)cc1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 1/20 0.46
HDAC6 Q9UBN7 4/20 0.43
HDAC1 Q13547 4/20 0.43
MAPT P10636 3/20 0.41
GAA P10253 1/20 0.41
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
KMT2A Q03164 1/20 0.40
SIRT2 Q8IXJ6 1/20 0.39
SIRT1 Q96EB6 1/20 0.39
TSHR P16473 1/20 0.39
TP53 P04637 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
NPC1 O15118 1/20 0.39
LMNA P02545 1/20 0.39
HTT P42858 1/20 0.39
HRH3 Q9Y5N1 2/20 0.39
MMP1 P03956 1/20 0.38
MMP13 P45452 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16321499 0.77 TDP1 (0.51) HDAC6MAPTTP53HTT
SCHEMBL29471237 0.73 GAA (0.46) HDAC6HDAC1MAPTGAAALDH1A1
SCHEMBL28825817 0.72 QPCTL (0.38) SLC22A12HDAC6HDAC1MAPTGAA
SCHEMBL28825821 0.71 NOTUM (0.44) MAPTMEN1KMT2ANPC1LMNA
SCHEMBL428976 0.71 GAA (0.44) MAPTGAAMEN1ALDH1A1KMT2A
SCHEMBL28050610 0.70 CDK5 (0.42) SLC22A12MAPTMEN1KMT2ANPC1
SCHEMBL16495396 0.70 ACHE (0.41) MAPTSIRT2SIRT1TSHRTP53
SCHEMBL16495185 0.68 CYP3A4 (0.39) MEN1ALDH1A1KMT2ATSHR
SCHEMBL447107 0.68 ACHE (0.50) MAPTMEN1KMT2AMMP1
SCHEMBL16321779 0.67 CPT1A (0.54) HDAC6MAPTTSHRTP53NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105308039-A Indolin-2-one or pyrrolo-pyridin/pyrimidin-2-one derivatives HOFFMANN LA ROCHE 2016-02-03 CN disclosed