SCHEMBL28825832

SCHEMBL28825832

N#Cc1c[c]ccc1Cc1ccc(-n2cccn2)cc1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MPO P05164 1/20 0.42
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
MAPK1 P28482 1/20 0.40
NOTUM Q6P988 1/20 0.40
DRD2 P14416 1/20 0.38
DRD4 P21917 1/20 0.38
DRD3 P35462 1/20 0.38
RORC P51449 4/20 0.38
CHRNA7 P36544 1/20 0.36
CHRNA10 Q9GZZ6 1/20 0.36
CHRNA9 Q9UGM1 1/20 0.36
CHRM1 P11229 5/20 0.36
NAMPT P43490 1/20 0.34
SCN9A Q15858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28050904 0.82 NOTUM (0.49) MPOKDM4EALDH1A1MAPK1NOTUM
SCHEMBL28093362 0.80 SMN1; SMN2 (0.41) KDM4EALDH1A1
SCHEMBL28093432 0.75 KDM4E (0.39) KDM4EALDH1A1MAPK1
SCHEMBL7237526 0.74 KDM4E (0.40) MPOKDM4EALDH1A1MAPK1NOTUM
SCHEMBL18725459 0.71 CHRM1 (0.48) MPOKDM4EALDH1A1MAPK1RORC
SCHEMBL27803014 0.71 KDM4E (0.44) MPOKDM4EALDH1A1MAPK1NOTUM
SCHEMBL11493922 0.70 NOTUM (0.53) MPOKDM4EALDH1A1MAPK1NOTUM
SCHEMBL18756219 0.70 MPO (0.45) MPOKDM4EALDH1A1MAPK1NOTUM
SCHEMBL41608 0.69 NOTUM (0.59) KDM4EALDH1A1MAPK1NOTUMDRD2
SCHEMBL18725387 0.69 CHRM1 (0.49) MPORORCCHRM1SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105209453-A Methylene linked quinolinyl modulators of ROR-gamma-T JANSSEN PHARMACEUTICA NV 2015-12-30 CN disclosed