SCHEMBL28050904

SCHEMBL28050904

Clc1c[c]ccc1Cc1ccc(-n2cccn2)cc1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.49
DRD2 P14416 1/20 0.45
DRD4 P21917 1/20 0.45
DRD3 P35462 1/20 0.45
MPO P05164 1/20 0.44
CHRM1 P11229 6/20 0.43
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPK1 P28482 1/20 0.42
DCTPP1 Q9H773 1/20 0.41
USP1 O94782 2/20 0.37
LMNA P02545 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
RORC P51449 3/20 0.36
CHRNA7 P36544 1/20 0.35
CHRNA10 Q9GZZ6 1/20 0.35
CHRNA9 Q9UGM1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28825832 0.82 MPO (0.42) NOTUMDRD2DRD4DRD3MPO
SCHEMBL18725397 0.74 NOTUM (0.49) NOTUMDRD2DRD4DRD3MPO
SCHEMBL7465412 0.73 CALM1 (0.41) ALDH1A1LMNASMN1; SMN2
SCHEMBL27803014 0.73 KDM4E (0.44) NOTUMDRD2DRD4DRD3MPO
SCHEMBL4878068 0.72 NOTUM (0.44) NOTUMKDM4EALDH1A1MAPK1LMNA
SCHEMBL41608 0.71 NOTUM (0.59) NOTUMDRD2DRD4DRD3CHRM1
SCHEMBL28181607 0.70 NOTUM (0.59) NOTUMDRD2DRD4DRD3MPO
SCHEMBL711055 0.70 NOTUM (0.63) NOTUMDRD2DRD4DRD3MPO
SCHEMBL28923071 0.70 KDM4E (0.46) NOTUMDRD2DRD4DRD3MPO
SCHEMBL1032919 0.69 NOTUM (0.53) NOTUMDRD2DRD4DRD3MPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105829294-A METHYLENE LINKED QUINOLINYL MODULATORS OF ROR-GAMMA-T 詹森药业有限公司 2016-08-03 CN disclosed
CN-105209453-A Methylene linked quinolinyl modulators of ROR-gamma-T JANSSEN PHARMACEUTICA NV 2015-12-30 CN disclosed