SCHEMBL28826568

SCHEMBL28826568

O=C(CCl)c1ccc(Br)c(C(F)(F)F)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.50
NPSR1 Q6W5P4 2/20 0.50
XBP1 P17861 1/20 0.50
HTT P42858 3/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
GSK3B P49841 5/20 0.47
LMNA P02545 3/20 0.47
NOTUM Q6P988 1/20 0.44
DDR1 Q08345 1/20 0.43
EPHX1 P07099 2/20 0.41
MAPK1 P28482 2/20 0.41
TRPA1 O75762 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HIF1A Q16665 1/20 0.41
TMPRSS4 Q9NRS4 1/20 0.41
GAA P10253 1/20 0.41
TAS2R14 Q9NYV8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5367304 0.86 GSK3B (0.47) MAPTRAB9AGSK3BNOTUMMAPK1
SCHEMBL7779146 0.84 PTPN1 (0.58) MAPTNPSR1XBP1HTTMEN1
SCHEMBL30580694 0.84 PTPN1 (0.58) MAPTNPSR1XBP1HTTMEN1
SCHEMBL5312305 0.83 TAS1R3 (0.49) GSK3BMAPK1TRPA1ALDH1A1HIF1A
SCHEMBL12097542 0.80 MAPT (0.54) MAPTNPSR1XBP1HTTMEN1
SCHEMBL6313753 0.80 PLOD2 (0.56) MAPTNPSR1XBP1HTTMEN1
SCHEMBL20714412 0.80 MAPT (0.48) MAPTNPSR1XBP1HTTMEN1
SCHEMBL20714414 0.80 MAPT (0.49) MAPTNPSR1XBP1HTTMEN1
SCHEMBL14419584 0.80 GSK3B (0.52) MAPTRAB9AGSK3BMAPK1TRPA1
SCHEMBL20703102 0.79 MAPT (0.47) MAPTNPSR1XBP1HTTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103415507-B As the 3-amino-pyridine class of GPBAR1 agonist HOFFMAN-LA ROCHE LTD. (CH) 2016-03-02 CN disclosed