SCHEMBL28827155

SCHEMBL28827155

O=[N+]([O-])c1cccc([CH]Br)c1F

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 1/20 0.47
TDP1 Q9NUW8 2/20 0.45
GPR35 Q9HC97 2/20 0.44
MAPT P10636 3/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
NPC1 O15118 1/20 0.41
MAPK1 P28482 1/20 0.41
RAB9A P51151 1/20 0.41
LMNA P02545 1/20 0.41
TSHR P16473 3/20 0.40
ALDH1A1 P00352 3/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
CA12 O43570 1/20 0.39
SOS1 Q07889 1/20 0.39
S100A4 P26447 1/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL698799 0.83 ERN1 (0.62) ERN1TDP1GPR35MAPTL3MBTL1
SCHEMBL12481825 0.81 ERN1 (0.47) ERN1TDP1GPR35MAPTL3MBTL1
SCHEMBL16952150 0.81 ERN1 (0.51) ERN1TDP1GPR35MAPTL3MBTL1
SCHEMBL2550458 0.80 MAPT (0.55) ERN1TDP1MAPTNPC1RAB9A
SCHEMBL3010961 0.80 TDP1 (0.61) ERN1TDP1GPR35TSHRALDH1A1
SCHEMBL7768221 0.79 ERN1 (0.49) ERN1TDP1GPR35MAPTL3MBTL1
SCHEMBL24492388 0.79 FBP1 (0.51) ERN1TDP1GPR35MAPTLMNA
SCHEMBL28704930 0.79 FBP1 (0.51) ERN1TDP1GPR35MAPTLMNA
Ammonia Solution, Strong SCHEMBL28763100 0.78 TDP1 (0.58) ERN1TDP1GPR35TSHRALDH1A1
SCHEMBL3073529 0.77 ERN1 (0.47) ERN1TDP1GPR35MAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104169283-B Fused quaternary or five-membered ring pyridophthalazinones as PARP inhibitors BEIGENE, LTD. (KY) 2016-05-18 CN disclosed