SCHEMBL28828583

SCHEMBL28828583

COc1ccc(-c2cc3c(cc2F)C(OC(N)=O)C(C)(C)C3)c(OC)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 2/20 0.38
MAP2K1 Q02750 2/20 0.38
DHODH Q02127 1/20 0.37
GRM2 Q14416 2/20 0.36
FFAR1 O14842 1/20 0.35
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35
TAS1R2 Q8TE23 1/20 0.35
CYP1A1 P04798 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2E1 P05181 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C8 P10632 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2A6 P11509 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP4B1 P13584 1/20 0.34
CYP2B6 P20813 1/20 0.34
CYP3A5 P20815 1/20 0.34
CYP2A7 P20853 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29121222 0.93 GRM2 (0.41) GRM2FFAR1SMN1; SMN2
SCHEMBL28828605 0.93 GRM2 (0.41) GRM2FFAR1SMN1; SMN2
SCHEMBL28828755 0.92 FFAR1 (0.37) GRM2FFAR1MEN1KMT2AADORA3
SCHEMBL28828713 0.92 GRM2 (0.39) DHODHGRM2SMN1; SMN2ERN1CYP19A1
SCHEMBL29121293 0.89 PRKAB2 (0.37) RAF1MAP2K1GRM2FFAR1TAS1R3
SCHEMBL28828507 0.89 PRKAB2 (0.37) RAF1MAP2K1GRM2FFAR1TAS1R3
SCHEMBL28828510 0.86 PRKAB2 (0.39) GRM2FFAR1CYP1A2CYP3A4CYP2D6
SCHEMBL29121219 0.86 PRKAB2 (0.39) GRM2FFAR1CYP1A2CYP3A4CYP2D6
SCHEMBL28828671 0.85 SLC9A1 (0.38) SMN1; SMN2MEN1KMT2AADORA3MAPT
SCHEMBL28828676 0.84 CYP1A1 (0.45) CYP1A1CYP1A2CYP2E1CYP3A4CYP2C8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114829361-B Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the same 柳韩洋行 2024-07-16 CN claimed
CN-114829361-A Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing same 柳韩洋行 2022-07-29 CN claimed
CN-114829361-B Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the same 柳韩洋行 2024-07-16 CN disclosed
CN-114829361-A Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing same 柳韩洋行 2022-07-29 CN disclosed