SCHEMBL28829286

SCHEMBL28829286

c1ccc(CCc2ccn(C(c3ccccc3)(c3ccccc3)c3ccccc3)n2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.43
KDM4A O75164 1/20 0.40
KDM5A P29375 1/20 0.40
KDM4C Q9H3R0 1/20 0.40
KDM5B Q9UGL1 1/20 0.40
EPHX2 P34913 1/20 0.38
NOS1 P29475 1/20 0.36
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
MAOB P27338 3/20 0.35
TAAR1 Q96RJ0 1/20 0.34
BACE1 P56817 2/20 0.34
MAOA P21397 2/20 0.33
PDE10A Q9Y233 1/20 0.33
HDAC1 Q13547 1/20 0.33
DAGLA Q9Y4D2 1/20 0.33
KCNN4 O15554 1/20 0.33
KCNA3 P22001 1/20 0.33
ESR1 P03372 1/20 0.33
ESR2 Q92731 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7969475 0.83 CYP4F2 (0.39) CYP11B1CYP11B2PDE10AHDAC1KCNN4
SCHEMBL5357402 0.81 P2RX7 (0.40) KCNH2CYP11B1CYP11B2MAOBMAOA
SCHEMBL5357577 0.79 CYP11B1 (0.37) KCNH2CYP11B1CYP11B2MAOBMAOA
SCHEMBL5361469 0.79 CYP11B1 (0.37) KCNH2CYP11B1CYP11B2MAOBMAOA
SCHEMBL10893727 0.75 IDO1 (0.37) CYP11B1CYP11B2KCNN4KCNA3
SCHEMBL6296621 0.74 CYP4F2 (0.36) HDAC1
SCHEMBL23646839 0.70 KCNH2 (0.47) KCNH2KDM4AKDM5AKDM4CKDM5B
SCHEMBL17356076 0.70 PDE10A (0.60) KCNH2KDM4AKDM5AKDM4CKDM5B
SCHEMBL15481206 0.70 ALPI (0.45)
SCHEMBL14478094 0.69 CYP11B1 (0.40) KCNH2NOS1CYP11B1CYP11B2MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105636586-A ERK inhibitors and methods of use ARAXES PHARMA LLC 2016-06-01 CN disclosed