SCHEMBL7969475

SCHEMBL7969475

OCCc1ccn(C(c2ccccc2)(c2ccccc2)c2ccccc2)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 1/20 0.39
CYP4A11 Q02928 1/20 0.39
TDP1 Q9NUW8 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
KCNN4 O15554 1/20 0.33
KCNA3 P22001 1/20 0.33
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32
HDAC1 Q13547 2/20 0.31
HDAC3 O15379 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC10 Q969S8 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
HDAC9 Q9UKV0 1/20 0.31
HDAC5 Q9UQL6 1/20 0.31
ACSS2 Q9NR19 1/20 0.31
PDE10A Q9Y233 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5357402 0.88 P2RX7 (0.40) CYP4F2CYP4A11TDP1CYP11B1CYP11B2
SCHEMBL28829286 0.83 KCNH2 (0.43) CYP11B1CYP11B2KCNN4KCNA3HDAC1
SCHEMBL27089076 0.80 EPHX2 (0.43)
SCHEMBL5357577 0.79 CYP11B1 (0.37) TDP1CYP11B1CYP11B2KCNN4KCNA3
SCHEMBL5361469 0.79 CYP11B1 (0.37) TDP1CYP11B1CYP11B2KCNN4KCNA3
SCHEMBL27087810 0.79 CYP11B1 (0.37) TDP1CYP11B1CYP11B2KCNN4KCNA3
SCHEMBL28221864 0.79 KCNN4 (0.37) TDP1CYP11B1CYP11B2KCNN4KCNA3
SCHEMBL6296621 0.77 CYP4F2 (0.36) CYP4F2CYP4A11HDAC1HDAC3HDAC2
SCHEMBL7986546 0.75 NOTUM (0.39) TDP1CA1CA2CA9
SCHEMBL10893727 0.75 IDO1 (0.37) CYP11B1CYP11B2KCNN4KCNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6174877-B1 EXCELLANT BACTERICIDES, ORAL ABSORBABILITY AND STABILITY; IMPROVE THE STABILITY TO RENAL DEHYDROPEPTIDASE I (DHP-I); 2-(2-(N-HETEROCYCLIC-ETHYLTHIO-) DERIVATIVES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-16 US disclosed
EP-0876370-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1998-11-11 EP disclosed
WO-1997025325-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-07-17 WO disclosed