SCHEMBL2883090

SCHEMBL2883090

COc1ccc(-c2cc(S(C)(=O)=O)ccc2Oc2cnn(C)c2)cn1

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.55
BRD4 O60885 6/20 0.44
PTGS1 P23219 1/20 0.43
PTGS2 P35354 1/20 0.43
FYN P06241 2/20 0.42
LOXL2 Q9Y4K0 2/20 0.41
SCN9A Q15858 2/20 0.41
OXTR P30559 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2224148 0.72 KCNH2 (1.00) KCNH2FYN
SCHEMBL16651342 0.71 BRD4 (0.68) BRD4
SCHEMBL28924973 0.71 PIK3CA (0.56) BRD4
SCHEMBL2226479 0.69 KCNH2 (0.90) KCNH2PTGS1PTGS2FYN
SCHEMBL562021 0.69 PIK3CD (0.58) KCNH2PTGS1PTGS2
SCHEMBL2227426 0.68 KCNH2 (0.78) KCNH2FYNOXTR
SCHEMBL6050909 0.67 PTGS2 (0.65) KCNH2PTGS1PTGS2FYNOXTR
SCHEMBL6050719 0.67 KCNH2 (0.63) KCNH2PTGS1PTGS2FYNOXTR
SCHEMBL30519619 0.67 CYP2A6 (0.50)
SCHEMBL1423797 0.67 CYP2A6 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059788-A1 PYRAZOLOPYRIDINE PI3K INHIBITOR COMPOUNDS AND METHODS OF USE GENENTECH, INC. (US) 2010-05-27 WO claimed