Caprolactam

Caprolactam

SCHEMBL28831685

CS(=O)(=O)O.O=C1CCCCCN1

nearest known ligand 0.67

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB2AGTR1BCL2BCL2A1BCL2L1BCL2L10BCL2L2BCRBRAFCHRM1CHRNA10CHRNA9DRD1DRD2DRD3DRD4DRD5EGFRF2FLT1FLT4GCKGHSRGNRHRGRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BHTR1AHTR1BHTR1DHTR2AHTR2CHTR3AIDH2KDRKITMAOBMCL1MTTPPP4HBPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PIKFYVEROCK1ROCK2SLC18A2SLC6A2SLC6A3SLC6A4TACR1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8gyrAgyrBparCparEpol

The experimentally established mechanism targets of Caprolactam. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 3/20 0.67
FKBP5 Q13451 1/20 0.67
OR51E2 Q9H255 1/20 0.56
KDM4E B2RXH2 2/20 0.47
GAA P10253 1/20 0.47
POLB P06746 1/20 0.47
MERTK Q12866 1/20 0.35
SIRT2 Q8IXJ6 4/20 0.35
SIRT1 Q96EB6 4/20 0.35
SIRT3 Q9NTG7 4/20 0.35
CCR2 P41597 3/20 0.34
CTSD P07339 5/20 0.34
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
2-Pyrrolidone SCHEMBL27503412 0.91 OR51E2 (0.68) CRBNFKBP5OR51E2KDM4EGAA
Caprolactam SCHEMBL1521129 0.91 CRBN (0.73) CRBNFKBP5OR51E2KDM4EGAA
Sulfuric Acid SCHEMBL28455727 0.91 CRBN (0.73) CRBNFKBP5OR51E2KDM4EGAA
Caprolactam SCHEMBL27823099 0.89 CRBN (0.70) CRBNFKBP5OR51E2KDM4EGAA
Caprolactam SCHEMBL27970597 0.89 CRBN (0.70) CRBNFKBP5OR51E2KDM4EGAA
Sulfuric Acid SCHEMBL30278662 0.89 CRBN (0.76) CRBNFKBP5OR51E2KDM4EGAA
Caprolactam SCHEMBL27842057 0.88 CRBN (0.67) CRBNFKBP5OR51E2KDM4EGAA
Caprolactam SCHEMBL10710154 0.87 CRBN (0.80) CRBNFKBP5OR51E2KDM4EGAA
Caprolactam SCHEMBL17238720 0.86 CRBN (0.64) CRBNFKBP5OR51E2KDM4EGAA
Caprolactam SCHEMBL28174316 0.84 CRBN (0.84) CRBNFKBP5OR51E2KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105669342-B A kind of method that p-tert-butyltoluene is synthesized using caprolactam class ionic liquid as catalyst 中国石油大学(华东) 2017-12-19 CN disclosed
CN-105669342-A Method of synthesizing p-tert-butyl toluene with caprolactam ionic liquid as catalyst 中国石油大学(华东) 2016-06-15 CN disclosed