SCHEMBL28832571

SCHEMBL28832571

Fc1cccc(NC2CC(F)(F)C2)n1

nearest known ligand 0.43

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 16/20 0.43
IDH2 P48735 5/20 0.43
CTSK P43235 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28085661 0.83 IDH1 (0.51) IDH1IDH2CTSK
SCHEMBL26618081 0.81 IDH1 (0.42) IDH1IDH2CTSK
SCHEMBL22547299 0.75 CTSK (0.42) CTSK
SCHEMBL17700614 0.74 GRM4 (0.45) IDH1IDH2
SCHEMBL26618136 0.73 GRM4 (0.39) IDH1IDH2
SCHEMBL15710124 0.70 IDH1 (0.36) IDH1IDH2
SCHEMBL21525591 0.70 HPGD (0.45) CTSK
SCHEMBL26618090 0.70 NOS2 (0.36) IDH1IDH2
SCHEMBL24065676 0.69 IDH1 (0.44) IDH1IDH2
SCHEMBL22547655 0.68 CTSK (0.34) CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102947305-B Compounds and methods for kinase modulation and indications therefor 普莱希科公司 2016-07-06 CN claimed
CN-102947305-B Compounds and methods for kinase modulation and indications therefor 普莱希科公司 2016-07-06 CN disclosed