SCHEMBL28832940

SCHEMBL28832940

CC(OC=O)c1ccc2c(ccn2COCC[Si](C)(C)C)c1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 5/20 0.33
NPC1 O15118 1/20 0.32
CYP19A1 P11511 2/20 0.32
HTR2A P28223 4/20 0.32
DGAT1 O75907 1/20 0.31
PPARG P37231 1/20 0.31
PPARD Q03181 1/20 0.31
PPARA Q07869 1/20 0.31
S1PR1 P21453 1/20 0.31
EGFR P00533 1/20 0.30
IGF1R P08069 1/20 0.30
SRC P12931 1/20 0.30
FLT4 P35916 1/20 0.30
KDR P35968 1/20 0.30
FLT3 P36888 1/20 0.30
EPHB4 P54760 1/20 0.30
TEK Q02763 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5744924 0.79 CYP2A6 (0.48) NPC1DGAT1EGFRIGF1RSRC
SCHEMBL28840671 0.76 HTR2C (0.48) HTR2CNPC1HTR2ADGAT1EGFR
SCHEMBL29925168 0.76 HTR2C (0.48) HTR2CNPC1HTR2ADGAT1EGFR
SCHEMBL4493915 0.74 HTR2C (0.49) HTR2CNPC1CYP19A1HTR2ADGAT1
SCHEMBL28840999 0.74 DGAT1 (0.36) HTR2CNPC1HTR2ADGAT1EGFR
SCHEMBL1467091 0.74 HTR2A (0.49) HTR2CNPC1HTR2ADGAT1
SCHEMBL29924680 0.74 DGAT1 (0.36) HTR2CNPC1HTR2ADGAT1EGFR
SCHEMBL29924782 0.74 HTR2C (0.49) HTR2CNPC1HTR2ADGAT1
SCHEMBL29924561 0.74 HTR2C (0.51) HTR2CHTR2A
SCHEMBL28840665 0.74 HTR2C (0.49) HTR2CNPC1HTR2ADGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105793252-A Inhibitors of bruton's tyrosine kinase 豪夫迈·罗氏有限公司 2016-07-20 CN disclosed