SCHEMBL28833101

SCHEMBL28833101

O=C(Oc1cccnc1)N1CCNc2ccccc21

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.44
AVPR1A P37288 1/20 0.44
HTR2C P28335 1/20 0.39
STAT3 P40763 1/20 0.39
KMT2A Q03164 3/20 0.39
ALOX15 P16050 1/20 0.39
ALDH1A1 P00352 2/20 0.38
POLB P06746 2/20 0.38
HSD17B10 Q99714 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
GPR6 P46095 1/20 0.38
GAA P10253 1/20 0.38
GPBAR1 Q8TDU6 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28092562 0.87 AVPR1A (0.49) HSD11B1AVPR1AKMT2AALDH1A1GAA
SCHEMBL28833120 0.80 AVPR1A (0.51) HSD11B1AVPR1AKMT2AALDH1A1MAPT
SCHEMBL28092466 0.80 BCHE (0.48) HSD11B1AVPR1AGPBAR1
SCHEMBL28092460 0.80 AVPR1A (0.45) HSD11B1AVPR1AKMT2AALOX15ALDH1A1
SCHEMBL28092473 0.79 BCHE (0.51) HSD11B1AVPR1AALDH1A1KDM4EGPBAR1
SCHEMBL28092698 0.79 BCHE (0.51) HSD11B1AVPR1AKMT2AALDH1A1MAPT
SCHEMBL28092682 0.79 AVPR1A (0.43) HSD11B1AVPR1AALOX15ALDH1A1GPR6
SCHEMBL28092668 0.77 MGLL (0.51) AVPR1AALDH1A1
SCHEMBL28092670 0.76 TRPV1 (0.46) AVPR1AKMT2AALDH1A1KDM4EMAPT
SCHEMBL28092729 0.76 MGLL (0.48) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106029076-A Benzopiperazine compositions as BET bromodomain inhibitors 福马疗法公司 2016-10-12 CN disclosed