SCHEMBL28833560

SCHEMBL28833560

CCc1c(N)cncc1Cl

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.40
CDK2 P24941 1/20 0.32
AOC3 Q16853 3/20 0.31
NOS3 P29474 1/20 0.31
NOS2 P35228 1/20 0.31
USP7 Q93009 2/20 0.31
PDE4D Q08499 4/20 0.31
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31
BDKRB2 P30411 1/20 0.30
ACP1 P24666 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10079575 0.84 PDE4D (0.35) GAAAOC3PDE4DPDE4APDE4B
SCHEMBL30937573 0.80 GAA (0.41) GAACDK2AOC3ACP1
SCHEMBL19986675 0.76 BDKRB2 (0.34) NOS3NOS2PDE4DPDE4APDE4B
SCHEMBL21736851 0.76 PDE4D (0.35) PDE4DPDE4APDE4BPDE4CBDKRB2
SCHEMBL24595059 0.74 CYP11B2 (0.34) AOC3NOS3NOS2USP7
SCHEMBL21736891 0.74 CYP11B2 (0.40) PDE4DPDE4APDE4BPDE4CBDKRB2
SCHEMBL20517931 0.74 AOC3 (0.31) AOC3NOS3NOS2
SCHEMBL24594992 0.74 PDE4D (0.31) PDE4DPDE4APDE4BPDE4CBDKRB2
SCHEMBL17681738 0.71 PDE4D (0.43) GAAPDE4DPDE4APDE4BPDE4C
SCHEMBL17366546 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105916503-A Heteroaryls and uses thereof 米伦纽姆医药公司 2016-08-31 CN disclosed