SCHEMBL28840246

SCHEMBL28840246

Cc1cc(C(C)C(=O)C(C)c2cc(C)c(OCC(F)F)c(C)c2)cc(C)c1OCC(F)F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN4A P35499 11/20 0.37
RXRA P19793 2/20 0.36
PPARG P37231 2/20 0.36
RARG P13631 1/20 0.36
RARB P10826 2/20 0.35
RARA P10276 1/20 0.35
RXRB P28702 1/20 0.35
RXRG P48443 1/20 0.35
LMNA P02545 2/20 0.34
SCN1A P35498 2/20 0.34
SCN5A Q14524 2/20 0.34
SCN9A Q15858 2/20 0.34
CYP1A2 P05177 2/20 0.34
CYP3A4 P08684 2/20 0.34
CYP2D6 P10635 2/20 0.34
NFKB1 P19838 2/20 0.34
CYP2C9 P11712 1/20 0.34
TSHR P16473 1/20 0.34
KCNK3 O14649 1/20 0.34
CACNA1F O60840 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27898774 0.85 SCN4A (0.38) SCN4ALMNASCN1ASCN5ASCN9A
SCHEMBL27986956 0.81 S1PR1 (0.43) CYP1A2TSHRGLAMAPT
SCHEMBL27931937 0.79 SCN9A (0.38) SCN9AMAPT
SCHEMBL4550431 0.78 SCN4A (0.46) SCN4ARXRAPPARGRARGLMNA
SCHEMBL28840247 0.77 SCN4A (0.37) SCN4ARXRAPPARGRARGRARB
SCHEMBL2714089 0.77 POLB (0.38) SCN4ARXRAPPARGRARGRARB
Hydrochloric Acid SCHEMBL2716056 0.77 SCN5A (0.46) SCN4ALMNASCN1ASCN5ASCN9A
SCHEMBL2716010 0.77 TPMT (0.39) SCN4ACYP1A2
SCHEMBL27986840 0.75 APP (0.38) PPARG
SCHEMBL19664495 0.75 GLA (0.47) SCN4ALMNASCN1ASCN5ASCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106478497-A Aryl amine derivatives as TTX S blocker 拉夸里亚创药株式会社 2017-03-08 CN disclosed