SCHEMBL28840472

SCHEMBL28840472

[CH2]C[C@@H](c1ccc([C@H](C)N)cc1)N1CCCCC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.45
CYP2C19 P33261 4/20 0.45
CYP3A4 P08684 3/20 0.45
CYP2D6 P10635 3/20 0.45
TSHR P16473 1/20 0.45
HRH3 Q9Y5N1 4/20 0.44
SLC6A2 P23975 3/20 0.42
SLC6A3 Q01959 3/20 0.42
SLC6A4 P31645 2/20 0.42
CYP2C9 P11712 3/20 0.40
HPGD P15428 1/20 0.40
MAPK1 P28482 1/20 0.40
ADRB2 P07550 1/20 0.39
ALDH1A1 P00352 1/20 0.38
TP53 P04637 1/20 0.37
POLB P06746 1/20 0.37
PKM P14618 1/20 0.36
KCNA5 P22460 2/20 0.36
KCNH2 Q12809 2/20 0.36
KCNE1 P15382 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28128634 1.00 CYP1A2 (0.45) CYP1A2CYP2C19CYP3A4CYP2D6TSHR
SCHEMBL28128314 0.80 CYP1A2 (0.41) CYP1A2CYP2C19CYP3A4CYP2D6TSHR
SCHEMBL28128317 0.80 CYP1A2 (0.41) CYP1A2CYP2C19CYP3A4CYP2D6TSHR
SCHEMBL28751840 0.80 TP53 (0.50) CYP1A2CYP2C19CYP3A4CYP2D6TSHR
SCHEMBL27585454 0.77 CYP1A2 (0.44) CYP1A2CYP2C19CYP3A4CYP2D6TSHR
Hydrochloric Acid SCHEMBL1935939 0.76 CYP2D6 (0.50) CYP1A2CYP2C19CYP3A4CYP2D6CYP2C9
SCHEMBL15797380 0.71 HRH3 (0.59) CYP1A2CYP2C19CYP3A4CYP2D6TSHR
SCHEMBL27548002 0.71 CYP1A2 (0.45) CYP1A2CYP2C19CYP3A4CYP2D6TSHR
SCHEMBL14831525 0.69 ALDH1A1 (0.55) CYP1A2CYP2C19CYP3A4HPGDMAPK1
SCHEMBL19601809 0.69 ALDH1A1 (0.55) CYP1A2CYP2C19CYP3A4HPGDMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106459008-A Phosphatidylinositol 3-kinase inhibitors 吉利德科学公司 2017-02-22 CN disclosed