SCHEMBL28844152

SCHEMBL28844152

COc1ccc(N(C(N)=O)c2ccccc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPM8 Q7Z2W7 2/20 0.56
KDM4E B2RXH2 1/20 0.54
HPGD P15428 1/20 0.54
KMT2A Q03164 2/20 0.51
TSHR P16473 2/20 0.51
MEN1 O00255 1/20 0.51
MTNR1A P48039 1/20 0.50
MTNR1B P49286 1/20 0.50
CES2 O00748 1/20 0.50
CES1 P23141 1/20 0.50
CA1 P00915 2/20 0.48
CA2 P00918 2/20 0.48
PARP1 P09874 1/20 0.48
PARP10 Q53GL7 1/20 0.48
PARP2 Q9UGN5 1/20 0.48
PARP4 Q9UKK3 1/20 0.48
PTGIR P43119 1/20 0.47
PTGDR Q13258 1/20 0.47
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL27597764 0.98 TRPM8 (0.55) TRPM8KDM4EHPGDKMT2ATSHR
SCHEMBL3470955 0.93 CA1 (0.55) TRPM8CES2CES1CA1CA2
SCHEMBL27515960 0.86 ESR2 (0.52) KMT2AMEN1CES2CES1CA1
SCHEMBL22204353 0.85 TRPM8 (0.59) TRPM8KDM4EHPGDKMT2ATSHR
SCHEMBL7616834 0.84 LMNA (0.50) TRPM8KDM4EHPGDKMT2ATSHR
SCHEMBL31393785 0.84 KMT2A (0.66) TRPM8KDM4EHPGDKMT2ATSHR
SCHEMBL5852226 0.83 ELANE (0.54) KDM4EKMT2ATSHRMEN1NPC1
Methyl Alcohol SCHEMBL28147253 0.82 NPSR1 (0.58) TRPM8HPGDKMT2ATSHRMEN1
SCHEMBL75883 0.82 NPSR1 (0.64) TRPM8HPGDKMT2ATSHRMEN1
SCHEMBL75885 0.82 NPSR1 (0.64) TRPM8HPGDKMT2ATSHRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104744356-B The synthetic method of 2-substituted carbamide class compound 上海大学 2017-05-31 CN disclosed