SCHEMBL28844196

SCHEMBL28844196

COc1ccc(-c2nc(Cn3cccc3)cs2)cc1.Cc1ccn(C)n1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.51
ALDH1A1 P00352 3/20 0.51
RAB9A P51151 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
HPGD P15428 2/20 0.48
ABCB1 P08183 2/20 0.47
ABCC1 P33527 1/20 0.47
ABCG2 Q9UNQ0 1/20 0.47
MAPT P10636 4/20 0.41
LMNA P02545 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
KLKB1 P03952 1/20 0.41
TP53 P04637 1/20 0.41
POLB P06746 1/20 0.40
ATM Q13315 1/20 0.40
HSD17B10 Q99714 1/20 0.40
F2RL3 Q96RI0 1/20 0.40
CYP19A1 P11511 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28294637 0.77 ALDH1A1 (0.47) KDM4EALDH1A1RAB9ATDP1HPGD
SCHEMBL5401821 0.75 KDM4E (0.56) KDM4EALDH1A1RAB9ATDP1HPGD
SCHEMBL28271026 0.73 DRD2 (0.63) KDM4EALDH1A1RAB9AHPGDMAPT
SCHEMBL28296211 0.73 KLKB1 (0.43) RAB9AKLKB1POLB
SCHEMBL28146146 0.72 KLKB1 (0.46) KDM4EALDH1A1HPGDMAPTLMNA
SCHEMBL5403605 0.71 KDM4E (0.56) KDM4EALDH1A1RAB9ATDP1HPGD
SCHEMBL201951 0.70 KDM4E (0.70) KDM4EALDH1A1RAB9ATDP1HPGD
SCHEMBL202826 0.70 KDM4E (0.70) KDM4EALDH1A1RAB9ATDP1HPGD
SCHEMBL3370261 0.70 KDM4E (0.97) KDM4EALDH1A1RAB9ATDP1HPGD
SCHEMBL2096148 0.69 MAPT (0.61) KDM4EALDH1A1RAB9ATDP1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106608872-A 5-pyrazole amide compound, and preparation method and application thereof 湖南化工研究院有限公司 2017-05-03 CN disclosed