SCHEMBL28844477

SCHEMBL28844477

COc1c(-c2ccccc2)nc2ccccc2c1C(=O)Nc1ccc(Oc2ccccc2)cc1

nearest known ligand 0.65

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 15/20 0.65
CYP3A4 P08684 2/20 0.58
TACR2 P21452 1/20 0.57
DHODH Q02127 1/20 0.53
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
GAA P10253 1/20 0.53
ADORA3 P0DMS8 1/20 0.49
KDM4E B2RXH2 1/20 0.49
LMNA P02545 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29864839 1.00 TACR3 (0.65) TACR3CYP3A4TACR2DHODHMEN1
SCHEMBL16098313 0.81 TACR3 (0.73) TACR3CYP3A4TACR2DHODH
SCHEMBL3963611 0.79 TACR3 (1.00) TACR3CYP3A4TACR2DHODH
SCHEMBL9199891 0.79 LMNA (0.60) CYP3A4MEN1KMT2AGAAADORA3
SCHEMBL3959255 0.78 TACR3 (0.68) TACR3CYP3A4TACR2DHODHLMNA
SCHEMBL3961862 0.76 TACR3 (0.67) TACR3CYP3A4TACR2DHODHLMNA
SCHEMBL8271391 0.76 TACR3 (0.65) TACR3CYP3A4TACR2DHODHLMNA
Ethane SCHEMBL6100955 0.74 TACR3 (0.54) TACR3CYP3A4TACR2MEN1KMT2A
SCHEMBL3959275 0.73 TACR3 (1.00) TACR3CYP3A4
SCHEMBL4895679 0.73 TACR3 (1.00) TACR3CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110105279-B Quinoline STAT3 specific inhibitor and preparation method and application thereof 中山大学 2022-09-16 CN disclosed