SCHEMBL28844538

SCHEMBL28844538

O=C(N1CCCC1c1ccc(Br)cc1)N1CCCC1c1ccc(Br)cc1

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CCNC P24863 1/20 0.51
CDK8 P49336 1/20 0.51
RIPK1 Q13546 2/20 0.49
SCD5 Q86SK9 2/20 0.47
HSD17B10 Q99714 1/20 0.43
HSP90AA1 P07900 1/20 0.43
HSP90AB1 P08238 1/20 0.43
TSHR P16473 1/20 0.42
AGTR2 P50052 2/20 0.41
CYP19A1 P11511 1/20 0.41
EPHX2 P34913 2/20 0.41
HSD11B1 P28845 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
MAPK1 P28482 1/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1423483 0.87 RIPK1 (0.50) CCNCCDK8RIPK1SCD5HSD17B10
SCHEMBL13300490 0.87 RIPK1 (0.50) CCNCCDK8RIPK1SCD5HSD17B10
SCHEMBL29515757 0.87 RIPK1 (0.50) CCNCCDK8RIPK1SCD5HSD17B10
SCHEMBL17453078 0.83 RIPK1 (0.47) CCNCCDK8RIPK1SCD5HSD17B10
SCHEMBL1778275 0.81 NR1H2 (0.53) CCNCCDK8RIPK1HSD17B10TSHR
SCHEMBL2169785 0.81 NR1H2 (0.53) CCNCCDK8RIPK1HSD17B10TSHR
SCHEMBL1778276 0.81 NR1H2 (0.53) CCNCCDK8RIPK1HSD17B10TSHR
SCHEMBL8957415 0.80 CCNC (0.46) CCNCCDK8RIPK1SCD5HSD17B10
SCHEMBL15300880 0.79 RIPK1 (0.47) CCNCCDK8RIPK1TSHRCYP2D6
SCHEMBL12650282 0.78 CCNC (0.43) CCNCCDK8RIPK1SCD5HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106817900-A Novel naphthyridines and isoquinolin and its purposes as CDK8/19 inhibitor 默克专利有限公司 2017-06-09 CN disclosed