SCHEMBL28844643

SCHEMBL28844643

NC(=O)c1cc2c(Br)ccc(F)c2[nH]1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 7/20 0.48
TDO2 P48775 7/20 0.48
MAP2K1 Q02750 1/20 0.47
HRH4 Q9H3N8 2/20 0.43
MAP2 P11137 1/20 0.39
DGAT1 O75907 1/20 0.38
RHEB Q15382 1/20 0.35
KIF11 P52732 1/20 0.35
NUDT1 P36639 1/20 0.34
GPR17 Q13304 1/20 0.33
BRD4 O60885 2/20 0.33
CCNC P24863 1/20 0.32
CDK8 P49336 1/20 0.32
EIF4A3 P38919 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29063246 0.89 MAP2K1 (0.49) IDO1TDO2MAP2K1HRH4MAP2
SCHEMBL29063177 0.88 IDO1 (0.54) IDO1TDO2MAP2K1HRH4MAP2
SCHEMBL22396294 0.85 IDO1 (0.65) IDO1TDO2HRH4RHEBGPR17
SCHEMBL20504672 0.81 IDO1 (0.48) IDO1TDO2MAP2K1HRH4MAP2
SCHEMBL29062921 0.81 IDO1 (0.48) IDO1TDO2MAP2K1HRH4MAP2
SCHEMBL22620603 0.80 XDH (0.50) IDO1TDO2HRH4
SCHEMBL20505200 0.77 KDM4E (0.57) IDO1TDO2HRH4BRD4
SCHEMBL30310687 0.77 KDM4E (0.57) IDO1TDO2HRH4BRD4
SCHEMBL28455876 0.77 ALOX15 (0.45) IDO1TDO2HRH4
SCHEMBL21724765 0.75 HRH4 (0.58) IDO1TDO2HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110483366-B Indole compound and preparation method, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2022-09-16 CN disclosed