SCHEMBL28845246

SCHEMBL28845246

[CH2]Cc1cc(C(C)C)[nH]n1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 2/20 0.44
HCAR3 P49019 1/20 0.44
PRKAB2 O43741 4/20 0.34
PRKAG1 P54619 4/20 0.34
PRKAA2 P54646 4/20 0.34
PRKAA1 Q13131 4/20 0.34
PRKAG3 Q9UGI9 4/20 0.34
PRKAG2 Q9UGJ0 4/20 0.34
PRKAB1 Q9Y478 4/20 0.34
TP53 P04637 3/20 0.33
MAPT P10636 3/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CCNA2 P20248 1/20 0.33
CDK2 P24941 1/20 0.33
CCNA1 P78396 1/20 0.33
KDM5A P29375 8/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1204783 0.81 HCAR2 (0.46) HCAR2HCAR3PRKAB2PRKAG1PRKAA2
SCHEMBL1206441 0.79 HCAR2 (0.44) HCAR2HCAR3PRKAB2PRKAG1PRKAA2
SCHEMBL12740609 0.79 HCAR2 (0.48) HCAR2HCAR3PRKAB2PRKAG1PRKAA2
SCHEMBL12775840 0.76 HCAR2 (0.42) HCAR2HCAR3PRKAB2PRKAG1PRKAA2
SCHEMBL1205832 0.75 HCAR2 (0.41) HCAR2HCAR3PRKAB2PRKAG1PRKAA2
SCHEMBL24622013 0.73 HPGD (0.44) HCAR2HCAR3TP53MAPTKDM5A
SCHEMBL27670323 0.71
SCHEMBL24622014 0.71 KCNH2 (0.43) HCAR2HCAR3TP53MAPTKDM5A
SCHEMBL28089341 0.69 HCAR2 (0.39) HCAR2HCAR3PRKAB2PRKAG1PRKAA2
SCHEMBL24622011 0.69 NOS3 (0.43) HCAR2HCAR3TP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106661043-A 2-oxa-5-azabicyclo[2.2.1]heptan-3-yl derivatives 豪夫迈·罗氏有限公司 2017-05-10 CN disclosed